SCHEMBL8810000

SCHEMBL8810000

CC(=O)Oc1ccc(Oc2cc(OCCc3ccc4ocnc4c3)ccc2C#N)cc1C

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.37
PDE4B Q07343 1/20 0.37
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
KMT2A Q03164 1/20 0.36
FNTA P49354 1/20 0.34
FNTB P49356 1/20 0.34
PGGT1B P53609 1/20 0.34
P2RX3 P56373 1/20 0.33
P2RX2 Q9UBL9 1/20 0.33
MRGPRX4 Q96LA9 1/20 0.33
AR P10275 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8810163 0.92 MRGPRX4 (0.41) MEN1ALDH1A1GAAKMT2AMRGPRX4
SCHEMBL8808406 0.85 MRGPRX4 (0.41) MRGPRX4
SCHEMBL8809995 0.78 MEN1 (0.43) MEN1ALDH1A1GAAKMT2AMRGPRX4
SCHEMBL8808917 0.75 XDH (0.45) FNTAFNTBPGGT1BMRGPRX4
SCHEMBL8809211 0.74 MAOB (0.54) MRGPRX4
SCHEMBL8814947 0.73 AR (0.40) PDE4BMEN1ALDH1A1GAAKMT2A
SCHEMBL8810273 0.73 MRGPRX4 (0.43) MRGPRX4
SCHEMBL8807149 0.73 NPC1 (0.48) MEN1KMT2AMRGPRX4
SCHEMBL8808922 0.72 FFAR1 (0.44) MRGPRX4
SCHEMBL8807665 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0805802-A1 SUBSTITUTED PHENYL COMPOUNDS AS ENDOTHELIN ANTAGONISTS RHONE-POULENC RORER LIMITED (GB) 1997-11-12 EP disclosed
WO-1996022978-A1 SUBSTITUTED PHENYL COMPOUNDS AS ENDOTHELIN ANTAGONISTS RHONE POULENC RORER LIMITED (GB) 1996-08-01 WO disclosed