SCHEMBL8811276

SCHEMBL8811276

O=C(Nc1ccc(F)cc1)c1cnoc1C(F)(F)F

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.58
SMN1; SMN2 Q16637 4/20 0.58
NPC1 O15118 4/20 0.58
LMNA P02545 3/20 0.58
CYP1A2 P05177 3/20 0.58
CYP2C9 P11712 3/20 0.58
HTT P42858 2/20 0.58
CYP2C19 P33261 2/20 0.58
GMNN O75496 1/20 0.58
TP53 P04637 1/20 0.58
CYP3A4 P08684 1/20 0.58
HTR1A P08908 1/20 0.58
THRB P10828 1/20 0.58
PIM1 P11309 1/20 0.58
MAOA P21397 1/20 0.58
SLC6A2 P23975 1/20 0.58
HTR2A P28223 1/20 0.58
AGTR1 P30556 1/20 0.58
CCKBR P32239 1/20 0.58
MC4R P32245 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11429607 0.89 DHODH (0.73) RAB9ASMN1; SMN2NPC1LMNACYP1A2
SCHEMBL8811957 0.87 LMNA (0.56) RAB9ASMN1; SMN2NPC1LMNACYP1A2
SCHEMBL8808712 0.83 MAPT (0.52) RAB9ASMN1; SMN2NPC1LMNACYP1A2
SCHEMBL11432410 0.83 NPC1 (0.65) RAB9ASMN1; SMN2NPC1LMNACYP1A2
SCHEMBL11441650 0.79 RAB9A (0.72) RAB9ASMN1; SMN2NPC1LMNACYP1A2
SCHEMBL9392605 0.78 PTPN1 (0.51) RAB9ASMN1; SMN2NPC1LMNACYP1A2
SCHEMBL9080725 0.78 NPC1 (0.53) RAB9ASMN1; SMN2NPC1HTTTP53
SCHEMBL8812402 0.76 DHODH (0.53) RAB9ASMN1; SMN2NPC1LMNACYP1A2
SCHEMBL8814086 0.75 KMT2A (0.55) RAB9ASMN1; SMN2NPC1LMNACYP1A2
SCHEMBL8809972 0.74 RAB9A (0.64) RAB9ASMN1; SMN2NPC1LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0527736-B1 ISOXAZOLE-4-CARBOXAMIDES AND HYDROXYALKYLIDENE-CYANOACETAMIDES, DRUGS CONTAINING THESE COMPOUNDS AND USE OF SUCH DRUGS HOECHST AG (DE) 1997-04-16 EP disclosed
US-5532259-A ANTITUMOR HOECHST AKTIENGESELLSCHAFT (DE) 1996-07-02 US disclosed
US-5494911-A TREATING LEUKEMIA, SARCOMA, CARCINOMA, LYMPHOMA, SKIN CANCER HOECHST AKTIENGESELLSCHAFT (DE) 1996-02-27 US disclosed