SCHEMBL8814869

SCHEMBL8814869

COc1cccc(-c2nc3c(-c4ccccc4)cccc3[nH]2)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.62
AURKA O14965 1/20 0.62
NR1I2 O75469 1/20 0.61
CYP1A2 P05177 1/20 0.61
VDR P11473 1/20 0.61
CYP2C9 P11712 1/20 0.61
CYP2B6 P20813 1/20 0.61
AHR P35869 1/20 0.61
NR1I3 Q14994 1/20 0.61
DHODH Q02127 3/20 0.54
NPC1 O15118 2/20 0.53
TP53 P04637 2/20 0.53
HPGD P15428 2/20 0.53
RAB9A P51151 2/20 0.53
KDM4E B2RXH2 1/20 0.53
ALDH1A1 P00352 1/20 0.53
TSHR P16473 1/20 0.53
NFKB1 P19838 1/20 0.53
NFKB2 Q00653 1/20 0.53
RELA Q04206 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8816887 0.92 PARP1 (0.53) PARP1AURKANR1I2CYP1A2VDR
SCHEMBL8814866 0.88 KDM4E (0.61) PARP1AURKACYP1A2DHODHNPC1
SCHEMBL4457030 0.85 DHODH (0.53) PARP1DHODHNPC1TP53HPGD
SCHEMBL8814874 0.84 PARP1 (0.63) PARP1DHODHTP53HPGDKDM4E
SCHEMBL230979 0.82 DHODH (0.53) PARP1CYP1A2DHODHNPC1RAB9A
SCHEMBL31027957 0.82 DHODH (0.59) PARP1CYP1A2DHODHNPC1RAB9A
SCHEMBL8817536 0.82 NR1I3 (0.58) PARP1NR1I3DHODHNPC1RAB9A
SCHEMBL8816555 0.82 DHODH (0.51) PARP1DHODHNPC1RAB9AMAPK14
SCHEMBL8818585 0.82 PARP1 (0.62) PARP1DHODHTP53HPGDKDM4E
SCHEMBL7146754 0.81 DHODH (0.62) PARP1CYP1A2DHODHNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997033873-A1 METHODS OF TREATING OR PREVENTING INTERSTITIAL CYSTITIS ELI LILLY AND COMPANY (US) 1997-09-18 WO disclosed
WO-1997031635-A1 METHODS OF TREATING OR PREVENTING SLEEP APNEA ELI LILLY AND COMPANY (US) 1997-09-04 WO disclosed