SCHEMBL8823947

SCHEMBL8823947

Cc1c([N+](=O)[O-])ccc2[nH]cc(CCCO)c12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 3/20 0.41
MTNR1A P48039 2/20 0.41
MTNR1B P49286 2/20 0.41
CHEK1 O14757 2/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
CDK1 P06493 1/20 0.35
CDK2 P24941 1/20 0.35
TXNRD1 Q16881 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MAPT P10636 2/20 0.35
RAD52 P43351 1/20 0.34
GPR84 Q9NQS5 1/20 0.34
PKM P14618 2/20 0.34
SLC6A4 P31645 1/20 0.33
TSHR P16473 1/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8824009 0.79 MEN1 (0.46) NQO2MTNR1AMTNR1BTDP1SMN1; SMN2
SCHEMBL18509788 0.79 GPR35 (0.41) NQO2MTNR1AMTNR1BCHEK1TDP1
SCHEMBL8823966 0.76 HTR2A (0.40) HTR2AHTR2CHTR2BSMN1; SMN2GPR84
SCHEMBL21378847 0.75 PTPRA (0.55) HTR2AHTR2CHTR2BMAPTSLC6A4
SCHEMBL21378848 0.75 PTPRA (0.55) HTR2AHTR2CHTR2BMAPTSLC6A4
SCHEMBL18508906 0.74 CDK2 (0.35) NQO2MTNR1AMTNR1BCHEK1CDK2
SCHEMBL25001171 0.70 HTR2C (0.51) NQO2MTNR1AMTNR1BHTR2AHTR2C
SCHEMBL4351496 0.70 NQO2 (0.64) NQO2HTR2AHTR2CCDK2SMN1; SMN2
SCHEMBL8824128 0.70 GLA (0.38) NQO2MTNR1AMTNR1BTDP1CDK1
SCHEMBL8978632 0.70 HTR2C (0.33) NQO2MTNR1AMTNR1BHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1063177-C Antimigraine 1,2,5-thiadiazole derivatives of indolylalkyl-pyridinyl and pyrimidinylpiperazines BRISTOL MYERS SQUIBB CO (US) 2001-03-14 CN disclosed
US-5618816-A Antimigraine 1,2,5-thiadiazole derivatives of indolylalkyl-pyridnyl and pyrimidinylpiperazines BRISTOL-MYERS SQUIBB COMPANY (US) 1997-04-08 US disclosed
CN-1138042-A Antimigraine 1,2,5-thiadiazole derivatives of indolylalkyl-pyridinyl and pyrimidinylpiperazines BRISTOL MYERS SQUIBB CO (US) 1996-12-18 CN disclosed
EP-0729958-A2 Antimigraine 1,2,5-thiadiazole derivatives of indolylalkyl-pyridinyl and pyrimidinyl-piperazines BRISTOL-MYERS SQUIBB COMPANY (US) 1996-09-04 EP disclosed
US-5521188-A Antimigraine cyclobutenedione derivatives of indolylalkyl-pyridinyl and pyrimidinylpiperazines BRISTOL-MYERS SQUIBB COMPANY (US) 1996-05-28 US disclosed
EP-0645385-A1 Antimigraine cyclobutenedione derivatives of indolylalkyl-pyridinyl and pyrimidinylpiperazines Bristol-Myers Squibb Company (US) 1995-03-29 EP disclosed