SCHEMBL8978632

SCHEMBL8978632

Cc1c(Nc2ccc3[nH]cc(CCCO)c3c2C)c(=O)c1=O

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 3/20 0.33
HTR2A P28223 2/20 0.33
HTR2B P41595 1/20 0.33
PTGS1 P23219 3/20 0.32
PARP1 P09874 1/20 0.32
KDM4E B2RXH2 2/20 0.32
MEN1 O00255 1/20 0.32
CYP2D6 P10635 1/20 0.32
KMT2A Q03164 1/20 0.32
SLC6A4 P31645 3/20 0.32
MPO P05164 3/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
GPR84 Q9NQS5 1/20 0.31
MTNR1A P48039 2/20 0.31
MTNR1B P49286 2/20 0.31
GFER P55789 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8978640 0.86
SCHEMBL8978715 0.82
SCHEMBL27456398 0.80 HTR2C (0.34) HTR2CHTR2AHTR2BKDM4EMEN1
SCHEMBL8627045 0.74 HTR2C (0.43) HTR2CHTR2AHTR2BKDM4EMEN1
SCHEMBL8823966 0.72 HTR2A (0.40) HTR2CHTR2AHTR2BCYP2D6SLC6A4
SCHEMBL8978742 0.71
SCHEMBL8978964 0.70 HTR1A (0.38) SLC6A4
SCHEMBL8823947 0.70 NQO2 (0.41) HTR2CHTR2AHTR2BMEN1KMT2A
SCHEMBL8629802 0.61 HTR1A (0.56) HTR2CHTR2AHTR2BCYP2D6KMT2A
SCHEMBL16540125 0.61 SLC6A4 (0.67) HTR2CHTR2AHTR2BSLC6A4GPR84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5521188-A Antimigraine cyclobutenedione derivatives of indolylalkyl-pyridinyl and pyrimidinylpiperazines BRISTOL-MYERS SQUIBB COMPANY (US) 1996-05-28 US disclosed
EP-0645385-A1 Antimigraine cyclobutenedione derivatives of indolylalkyl-pyridinyl and pyrimidinylpiperazines Bristol-Myers Squibb Company (US) 1995-03-29 EP disclosed