SCHEMBL8824092

SCHEMBL8824092

ON=C1CCn2c(-c3ccc(Br)cc3)nc3cccc1c32

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 14/20 0.45
GRM2 Q14416 4/20 0.38
HTR3A P46098 1/20 0.37
KCNH2 Q12809 3/20 0.35
KDM4E B2RXH2 1/20 0.35
RECQL P46063 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8824089 1.00 PARP1 (0.45) PARP1GRM2HTR3AKCNH2KDM4E
SCHEMBL9243355 0.89 PARP1 (0.55) PARP1GRM2HTR3AKCNH2KDM4E
SCHEMBL8824093 0.89 PARP1 (0.55) PARP1GRM2HTR3AKCNH2KDM4E
SCHEMBL8823991 0.88 PARP1 (0.58) PARP1GRM2HTR3AKCNH2KDM4E
SCHEMBL8823994 0.88 PARP1 (0.58) PARP1GRM2HTR3AKCNH2KDM4E
SCHEMBL8824085 0.85 PARP1 (0.47) PARP1GRM2HTR3AKCNH2KDM4E
SCHEMBL8824082 0.85 PARP1 (0.47) PARP1GRM2HTR3AKCNH2KDM4E
SCHEMBL8824037 0.83 PARP1 (0.42) PARP1GRM2HTR3AKCNH2KDM4E
SCHEMBL8824032 0.83 PARP1 (0.42) PARP1GRM2HTR3AKCNH2KDM4E
SCHEMBL9036918 0.79 ALDH1A1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5643920-A PYRROLO(3,2,1-IJ)QUINOLINES MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1997-07-01 US disclosed
EP-0638570-A1 TRICYCLIC COMPOUND HAVING ANTIALLERGIC EFFECT MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1995-02-15 EP disclosed