SCHEMBL8825554

SCHEMBL8825554

CCNc1cc2ncnc(NCc3ccc(F)cc3)c2cc1[N+](=O)[O-]

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 8/20 0.57
ERBB2 P04626 3/20 0.57
USP10 Q14694 1/20 0.56
PIK3C3 Q8NEB9 1/20 0.56
USP13 Q92995 1/20 0.56
HTT P42858 2/20 0.51
CNR1 P21554 1/20 0.46
CNR2 P34972 1/20 0.46
LMNA P02545 1/20 0.46
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
HDAC9 Q9UKV0 1/20 0.44
HDAC5 Q9UQL6 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7524564 0.91 EGFR (0.50) EGFRERBB2USP10PIK3C3USP13
SCHEMBL8825884 0.91 ALDH1A1 (0.55) EGFRERBB2HTTLMNAKDM4E
SCHEMBL8825593 0.90 EGFR (0.46) EGFRERBB2USP10PIK3C3USP13
SCHEMBL8825977 0.90 MAPK1 (0.55) EGFRERBB2HTTCNR1CNR2
SCHEMBL8795709 0.90 EGFR (0.49) EGFRERBB2HTTKDM4EALDH1A1
SCHEMBL8825839 0.89 EGFR (0.62) EGFRHTTLMNAKDM4E
SCHEMBL7522588 0.89 EGFR (0.47) EGFRERBB2USP10PIK3C3USP13
SCHEMBL7521999 0.89 EGFR (0.50) EGFRERBB2USP10PIK3C3USP13
SCHEMBL8825848 0.88 EGFR (0.50) EGFRERBB2HTTLMNAKDM4E
SCHEMBL8825757 0.88 KDM4E (0.51) EGFRERBB2HTTLMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5661147-A CYCLIC GUANOSINE MONOPHOSPHATE-SPECIFIC PHOSPHODIESTERASE INHIBITOR; TREATING CARDIOVASCULAR DISORDER KYOWA HAKKO KOGYO CO., LTD. (JP) 1997-08-26 US disclosed
EP-0668280-A1 IMIDAZOQUINAZOLINE DERIVATIVE KYOWA HAKKO KOGYO CO., LTD. (JP) 1995-08-23 EP disclosed