SCHEMBL8827591

SCHEMBL8827591

O=C(c1ccc([N+](=O)[O-])nc1)N1CCCCc2cc(Cl)ccc21

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 7/20 0.60
HDAC1 Q13547 2/20 0.54
HDAC6 Q9UBN7 2/20 0.54
AVPR1A P37288 3/20 0.51
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
ALDH1A1 P00352 2/20 0.47
IDO1 P14902 3/20 0.46
KCNH2 Q12809 3/20 0.46
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
CA14 Q9ULX7 1/20 0.43
MAPT P10636 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
OXTR P30559 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8827616 0.84 HDAC1 (0.43) AVPR2HDAC1HDAC6AVPR1AMEN1
SCHEMBL8827667 0.84 LMNA (0.43) AVPR2HDAC1HDAC6AVPR1AMEN1
SCHEMBL8827639 0.83 AVPR2 (0.65) AVPR2HDAC1HDAC6AVPR1AALDH1A1
SCHEMBL8827571 0.82 AVPR1A (0.41) AVPR2HDAC1HDAC6AVPR1AMEN1
SCHEMBL8827659 0.79 AVPR2 (0.38) AVPR2HDAC1HDAC6AVPR1AMEN1
SCHEMBL30824934 0.75 AVPR2 (0.70) AVPR2HDAC1HDAC6AVPR1AALDH1A1
SCHEMBL8827653 0.74 AVPR2 (0.33) AVPR2HDAC1HDAC6AVPR1AMEN1
SCHEMBL8827601 0.74 AVPR2 (0.36) AVPR2HDAC1HDAC6AVPR1AMEN1
SCHEMBL8827637 0.74 PTGDR (0.39) AVPR2HDAC1HDAC6AVPR1AMEN1
SCHEMBL7240942 0.73 AVPR2 (0.69) AVPR2HDAC1HDAC6AVPR1AIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5677299-A VASOPRESSIN OR OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1997-10-14 US disclosed
US-5498609-A Benzoazepinyl compounds as oxytocin and vasopressin antagonists OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1996-03-12 US disclosed
EP-0612319-A1 BENZOHETEROCYCLIC COMPOUNDS AS OXYTOCIN AND VASOPRESSIN ANTAGONISTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-08-31 EP disclosed
WO-1994004525-A1 BENZOHETEROCYCLIC COMPOUNDS AS OXYTOCIN AND VASOPRESSIN ANTAGONISTS OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1994-03-03 WO disclosed