SCHEMBL8828215

SCHEMBL8828215

COc1ccc(CCN(C)CCCN(C(=O)C/C=C/c2ccc(C#N)cc2)C2CCCC2)cc1OC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 8/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2D6 P10635 2/20 0.41
PMP22 Q01453 2/20 0.41
BLM P54132 1/20 0.41
SMPD1 P17405 1/20 0.40
CYP2C19 P33261 4/20 0.40
CYP2C9 P11712 3/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
ALDH1A1 P00352 1/20 0.40
ABCB1 P08183 6/20 0.39
ABCC1 P33527 3/20 0.39
MAPT P10636 3/20 0.39
KCNH2 Q12809 3/20 0.39
ABCB11 O95342 2/20 0.39
SCN1A P35498 2/20 0.39
SCN2A Q99250 2/20 0.39
SCN3A Q9NY46 2/20 0.39
TSHR P16473 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8828132 0.90 MAPT (0.44) CYP3A4CYP1A2CYP2D6PMP22BLM
SCHEMBL8828377 0.90 CYP3A4 (0.50) CYP3A4CYP1A2CYP2D6PMP22BLM
SCHEMBL8828424 0.89 SMPD1 (0.50) CYP3A4CYP1A2CYP2D6PMP22BLM
SCHEMBL8828159 0.84 HTR2A (0.47) HTR1AADRA2ADRD2ADRA2BADRA2C
SCHEMBL8828359 0.83 KMT2A (0.39) CYP3A4CYP1A2CYP2D6PMP22BLM
SCHEMBL8828339 0.82 KMT2A (0.38) CYP3A4CYP1A2CYP2D6PMP22BLM
SCHEMBL8828260 0.80 OPRM1 (0.47) CYP3A4CYP1A2CYP2D6PMP22BLM
SCHEMBL8828234 0.75 CYP3A4 (0.50) CYP3A4CYP1A2CYP2D6PMP22BLM
SCHEMBL8828430 0.75 MAPT (0.59) MEN1KMT2AALDH1A1MAPTLMNA
SCHEMBL8828400 0.73 CYP3A4 (0.47) CYP3A4CYP1A2CYP2D6PMP22BLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607953-A ANTIISCHEMIC AGENTS EISAI CO., LTD. (JP) 1997-03-04 US disclosed
EP-0344577-B1 Butenoic or propenoic acid derivatives EISAI CO LTD (JP) 1996-10-09 EP disclosed
US-5382595-A Antiischemic agents EISAI CO., LTD. (JP) 1995-01-17 US disclosed
US-5177089-A Antiischemic agent, vasodilator EISAI CO., LTD. (JP) 1993-01-05 US disclosed
US-5047417-A Butenoic or propenoic acid derivatives EISAI CO. LTD. (JP) 1991-09-10 US disclosed
EP-0344577-A2 Butenoic or propenoic acid derivatives Eisai Co., Ltd. (JP) 1989-12-06 EP disclosed