SCHEMBL8828339

SCHEMBL8828339

COc1ccc(CCN(C)CCCN(C(=O)C/C=C/c2ccc(-n3ccnc3C)cc2)C2CCCC2)cc1OC

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.38
ALDH1A1 P00352 5/20 0.38
LMNA P02545 1/20 0.38
ABCB1 P08183 1/20 0.37
SMPD1 P17405 3/20 0.37
MAPT P10636 2/20 0.37
HCN4 Q9Y3Q4 1/20 0.37
CYP3A4 P08684 4/20 0.37
MEN1 O00255 3/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
HSP90AA1 P07900 1/20 0.37
CTSD P07339 1/20 0.36
ALOX15 P16050 1/20 0.36
BLM P54132 1/20 0.36
PMP22 Q01453 1/20 0.36
KDM4E B2RXH2 1/20 0.36
POLB P06746 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8828359 0.86 KMT2A (0.39) KMT2AALDH1A1ABCB1SMPD1MAPT
SCHEMBL8828132 0.86 MAPT (0.44) KMT2AALDH1A1SMPD1MAPTHCN4
SCHEMBL8828377 0.85 CYP3A4 (0.50) KMT2AALDH1A1LMNASMPD1MAPT
SCHEMBL8828424 0.84 SMPD1 (0.50) KMT2AALDH1A1LMNAABCB1SMPD1
SCHEMBL8828158 0.82 OPRM1 (0.44) KMT2AALDH1A1LMNAABCB1SMPD1
SCHEMBL8828215 0.82 CYP3A4 (0.41) KMT2AALDH1A1LMNAABCB1SMPD1
SCHEMBL8828159 0.79 HTR2A (0.47)
SCHEMBL8828232 0.74 ALDH1A1 (0.42) KMT2AALDH1A1LMNASMPD1MAPT
SCHEMBL8828234 0.71 CYP3A4 (0.50) KMT2AALDH1A1LMNAABCB1SMPD1
SCHEMBL9233122 0.69 OPRM1 (0.42) KMT2AALDH1A1MAPTCYP3A4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607953-A ANTIISCHEMIC AGENTS EISAI CO., LTD. (JP) 1997-03-04 US disclosed
EP-0344577-B1 Butenoic or propenoic acid derivatives EISAI CO LTD (JP) 1996-10-09 EP disclosed
US-5382595-A Antiischemic agents EISAI CO., LTD. (JP) 1995-01-17 US disclosed
US-5177089-A Antiischemic agent, vasodilator EISAI CO., LTD. (JP) 1993-01-05 US disclosed
EP-0344577-A2 Butenoic or propenoic acid derivatives Eisai Co., Ltd. (JP) 1989-12-06 EP disclosed