SCHEMBL8828293

SCHEMBL8828293

CC(C)N(CCCN)CCc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.50
AOC3 Q16853 4/20 0.49
SIGMAR1 Q99720 3/20 0.47
TAAR1 Q96RJ0 2/20 0.46
HTR2A P28223 2/20 0.45
CYP2A6 P11509 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
LOXL2 Q9Y4K0 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19129470 0.87 TAAR1 (0.58) AOC3SIGMAR1TAAR1
SCHEMBL3874218 0.84 SIGMAR1 (0.53) MAOAAOC3SIGMAR1HTR2ASMN1; SMN2
Hydrochloric Acid SCHEMBL31687522 0.83 SIGMAR1 (0.51) MAOAAOC3SIGMAR1HTR2ASMN1; SMN2
SCHEMBL14065247 0.80 TAAR1 (0.50) AOC3SIGMAR1TAAR1
SCHEMBL9114952 0.79 ALDH1A1 (0.49) AOC3SIGMAR1TAAR1HTR2ASMN1; SMN2
SCHEMBL26239740 0.79 AOC3 (0.56) AOC3SIGMAR1TAAR1
SCHEMBL26243215 0.77 SIGMAR1 (0.57) AOC3SIGMAR1
SCHEMBL8179163 0.77 AOC3 (0.54) MAOAAOC3SIGMAR1TAAR1CYP2A6
SCHEMBL9459857 0.77 CHRM2 (0.38)
SCHEMBL14064920 0.77 AOC3 (0.62) AOC3SIGMAR1TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607953-A ANTIISCHEMIC AGENTS EISAI CO., LTD. (JP) 1997-03-04 US disclosed
EP-0344577-B1 Butenoic or propenoic acid derivatives EISAI CO LTD (JP) 1996-10-09 EP disclosed
US-5382595-A Antiischemic agents EISAI CO., LTD. (JP) 1995-01-17 US disclosed
US-5177089-A Antiischemic agent, vasodilator EISAI CO., LTD. (JP) 1993-01-05 US disclosed
US-5047417-A Butenoic or propenoic acid derivatives EISAI CO. LTD. (JP) 1991-09-10 US disclosed
CN-1040366-A Butenoic acid or acrylic acid derivative EISAI CO LTD (JP) 1990-03-14 CN disclosed
EP-0344577-A2 Butenoic or propenoic acid derivatives Eisai Co., Ltd. (JP) 1989-12-06 EP disclosed