SCHEMBL8828367

SCHEMBL8828367

COc1ccc(OC)c(CCN(C)CCCNC(=O)C/C=C/c2ccc(-n3ccnc3)cc2)c1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41
DRD3 P35462 2/20 0.40
DRD2 P14416 1/20 0.40
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
GAA P10253 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8828318 0.89 DRD3 (0.44) DRD3DRD2CYP11B1CYP11B2GAA
SCHEMBL8828195 0.88 OPRM1 (0.44) GAA
SCHEMBL8828202 0.88 DRD3 (0.41) DRD3DRD2CYP11B1CYP11B2GAA
Hydrochloric Acid SCHEMBL6368810 0.88 DRD3 (0.41) DRD3DRD2CYP11B1CYP11B2GAA
SCHEMBL8828419 0.87 MAOB (0.38) DRD3DRD2
SCHEMBL8828168 0.87 DRD3 (0.45) MTNR1AMTNR1BDRD3DRD2
SCHEMBL9231352 0.87 DRD3 (0.45) DRD3DRD2CYP11B1CYP11B2GAA
SCHEMBL9233122 0.86 OPRM1 (0.42) GAA
SCHEMBL9155730 0.86 DRD3 (0.42) DRD3DRD2CYP11B1CYP11B2GAA
SCHEMBL9160192 0.85 CYP3A4 (0.38) DRD3DRD2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607953-A ANTIISCHEMIC AGENTS EISAI CO., LTD. (JP) 1997-03-04 US disclosed
EP-0344577-B1 Butenoic or propenoic acid derivatives EISAI CO LTD (JP) 1996-10-09 EP disclosed
US-5382595-A Antiischemic agents EISAI CO., LTD. (JP) 1995-01-17 US disclosed
US-5177089-A Antiischemic agent, vasodilator EISAI CO., LTD. (JP) 1993-01-05 US disclosed
EP-0344577-A2 Butenoic or propenoic acid derivatives Eisai Co., Ltd. (JP) 1989-12-06 EP disclosed