SCHEMBL8828419

SCHEMBL8828419

COc1cc(CCN(C)CCCNC(=O)C/C=C/c2ccc(-n3ccnc3)cc2)cc(OC)c1OC

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.38
DRD3 P35462 4/20 0.38
DRD2 P14416 3/20 0.38
CYP24A1 Q07973 1/20 0.38
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.37
PKM P14618 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
HTT P42858 1/20 0.36
OPRM1 P35372 1/20 0.36
TMEM97 Q5BJF2 1/20 0.36
SIGMAR1 Q99720 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8828195 0.92 OPRM1 (0.44) MAOBALDH1A1KDM4EPKMMEN1
SCHEMBL8828202 0.91 DRD3 (0.41) MAOBDRD3DRD2
SCHEMBL9233122 0.90 OPRM1 (0.42) MAOBALDH1A1KDM4EMEN1KMT2A
Hydrochloric Acid SCHEMBL6368810 0.90 DRD3 (0.41) MAOBDRD3DRD2
SCHEMBL9155730 0.88 DRD3 (0.42) MAOBDRD3DRD2
SCHEMBL8828318 0.88 DRD3 (0.44) MAOBDRD3DRD2ALDH1A1
SCHEMBL8828168 0.88 DRD3 (0.45) DRD3DRD2KDM4ESIGMAR1
SCHEMBL9160192 0.87 CYP3A4 (0.38) MAOBDRD3DRD2ALDH1A1KDM4E
SCHEMBL8828367 0.87 MTNR1A (0.41) DRD3DRD2
SCHEMBL9160628 0.86 MAOB (0.38) MAOBDRD3DRD2OPRM1TMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0344577-B1 Butenoic or propenoic acid derivatives EISAI CO LTD (JP) 1996-10-09 EP claimed
US-5607953-A ANTIISCHEMIC AGENTS EISAI CO., LTD. (JP) 1997-03-04 US disclosed
EP-0344577-B1 Butenoic or propenoic acid derivatives EISAI CO LTD (JP) 1996-10-09 EP disclosed
US-5382595-A Antiischemic agents EISAI CO., LTD. (JP) 1995-01-17 US disclosed
US-5177089-A Antiischemic agent, vasodilator EISAI CO., LTD. (JP) 1993-01-05 US disclosed
US-5047417-A Butenoic or propenoic acid derivatives EISAI CO. LTD. (JP) 1991-09-10 US disclosed
EP-0344577-A2 Butenoic or propenoic acid derivatives Eisai Co., Ltd. (JP) 1989-12-06 EP disclosed