SCHEMBL8828375

SCHEMBL8828375

O=C(O)CC=Cc1ccc(-c2ccccn2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PAM P19021 1/20 0.60
HDAC1 Q13547 3/20 0.47
HDAC3 O15379 2/20 0.47
HDAC2 Q92769 2/20 0.47
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
MAPT P10636 2/20 0.44
KDM4E B2RXH2 1/20 0.44
LMNA P02545 1/20 0.44
PKM P14618 1/20 0.44
DHODH Q02127 1/20 0.44
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
MAOB P27338 1/20 0.41
HCAR2 Q8TDS4 1/20 0.41
CA12 O43570 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8828368 1.00 PAM (0.60) PAMHDAC1HDAC3HDAC2NPC1
SCHEMBL6852650 0.83 HDAC3 (0.46) HDAC1HDAC3HDAC2NPC1RAB9A
SCHEMBL6852658 0.83 HDAC3 (0.46) HDAC1HDAC3HDAC2NPC1RAB9A
SCHEMBL10942613 0.81 PAM (0.78) PAMHDAC1HDAC3HDAC2RAB9A
SCHEMBL10942618 0.81 PAM (0.78) PAMHDAC1HDAC3HDAC2RAB9A
SCHEMBL10942607 0.81 PAM (0.78) PAMHDAC1HDAC3HDAC2RAB9A
SCHEMBL11827477 0.80 HDAC2 (0.56) HDAC1HDAC3HDAC2NPC1RAB9A
SCHEMBL11827474 0.80 HDAC2 (0.56) HDAC1HDAC3HDAC2NPC1RAB9A
SCHEMBL13017261 0.79 KDM4E (0.50) HDAC1HDAC3HDAC2NPC1RAB9A
SCHEMBL582727 0.77 PAM (1.00) PAMHDAC1HDAC3HDAC2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607953-A ANTIISCHEMIC AGENTS EISAI CO., LTD. (JP) 1997-03-04 US disclosed
EP-0344577-B1 Butenoic or propenoic acid derivatives EISAI CO LTD (JP) 1996-10-09 EP disclosed
US-5382595-A Antiischemic agents EISAI CO., LTD. (JP) 1995-01-17 US disclosed
US-5177089-A Antiischemic agent, vasodilator EISAI CO., LTD. (JP) 1993-01-05 US disclosed
EP-0344577-A2 Butenoic or propenoic acid derivatives Eisai Co., Ltd. (JP) 1989-12-06 EP disclosed