SCHEMBL8828527

SCHEMBL8828527

CN(C)C(=O)c1cc(C#N)cnc1Cl

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIK3C3 Q8NEB9 1/20 0.45
ALDH1A1 P00352 1/20 0.37
F10 P00742 1/20 0.36
TMPRSS4 Q9NRS4 1/20 0.36
CNR1 P21554 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
PDPK1 O15530 1/20 0.35
KMT2A Q03164 1/20 0.35
MTOR P42345 2/20 0.35
CCNE1 P24864 1/20 0.35
CDK2 P24941 1/20 0.35
LRRK2 Q5S007 1/20 0.35
S1PR1 P21453 1/20 0.35
S1PR3 Q99500 1/20 0.35
AR P10275 1/20 0.35
PPARG P37231 1/20 0.34
CDK1 P06493 1/20 0.34
CHEK1 O14757 1/20 0.34
IRAK4 Q9NWZ3 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8931160 0.78 PIK3C3 (0.50) PIK3C3ALDH1A1F10CNR1KMT2A
SCHEMBL31108710 0.78 KDM4E (0.41) ALDH1A1TMPRSS4TDP1KMT2APPARG
SCHEMBL8828399 0.77 PIK3C3 (0.49) PIK3C3ALDH1A1CNR1KMT2AMTOR
SCHEMBL15999462 0.76 ALDH1A1 (0.56) PIK3C3ALDH1A1CNR1KMT2ALRRK2
SCHEMBL22890272 0.76 LRRK2 (0.40) ALDH1A1TMPRSS4TDP1LRRK2AR
SCHEMBL8828590 0.76 PIK3C3 (0.48) PIK3C3ALDH1A1CNR1KMT2ALRRK2
SCHEMBL8548977 0.73 PIK3C3 (0.46) PIK3C3ALDH1A1CNR1KMT2ALRRK2
SCHEMBL8828506 0.71 PIK3C3 (0.41) PIK3C3ALDH1A1CNR1KMT2A
SCHEMBL30033113 0.71 FLT1 (0.48) ALDH1A1MTORCCNE1CDK2AR
SCHEMBL13943063 0.69 EGLN1 (0.40) ALDH1A1CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5688795-A URINARY TRACTS OBSTRUCTION SYNTEX (U.S.A.) INC. (US) 1997-11-18 US disclosed
EP-0711757-A1 3-(4-phenylpiperazin-1-yl)propyl-amino, thio and oxy -pyridine, pyrimidine and benzene derivatives as alpha1-adrenoceptor antagonists F. Hoffmann-La Roche AG (CH) 1996-05-15 EP disclosed