SCHEMBL883040

SCHEMBL883040

COc1ccc2c(O[C@@H]3C[C@@H](C(N)=O)N(C(=O)OC(C)(C)C)C3)cc(-c3nc(C(C)C)cs3)nc2c1C

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.43
UCHL1 P09936 1/20 0.37
CTSB P07858 1/20 0.35
PPP3CB P16298 1/20 0.35
ADRB3 P13945 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34
PDE4B Q07343 8/20 0.34
PDE4A P27815 2/20 0.32
PDE4C Q08493 2/20 0.32
PDE4D Q08499 2/20 0.32
HTRA1 Q92743 1/20 0.31
PIK3CD O00329 2/20 0.31
PIK3CA P42336 2/20 0.31
PIK3CB P42338 2/20 0.31
PIK3CG P48736 2/20 0.31
MCL1 Q07820 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1101734 0.94 CTSS (0.44) CTSSUCHL1CTSBPPP3CBADRB3
SCHEMBL7936436 0.94 CTSS (0.44) CTSSUCHL1CTSBPPP3CBADRB3
SCHEMBL1101688 0.93 CTSS (0.44) CTSSUCHL1CTSBPPP3CBADRB3
SCHEMBL12775112 0.86 UCHL1 (0.38) CTSSUCHL1CTSBPPP3CBADRB3
SCHEMBL313204 0.86 UCHL1 (0.38) CTSSUCHL1CTSBPPP3CBPDE4B
SCHEMBL1101736 0.86 UCHL1 (0.38) CTSSUCHL1CTSBPPP3CBPDE4B
SCHEMBL2213932 0.86 UCHL1 (0.38) CTSSUCHL1CTSBPPP3CBPDE4B
SCHEMBL312697 0.85 CTSS (0.38) CTSSUCHL1CTSBPPP3CBPDE4B
SCHEMBL312698 0.85 CTSS (0.38) CTSSUCHL1CTSBPPP3CBPDE4B
SCHEMBL882935 0.85 CTSS (0.39) CTSSPDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012040242-A1 SUBSTITUTED PROLINE INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2012-03-29 WO disclosed