SCHEMBL8830945

SCHEMBL8830945

IC1=CCN(Cc2ccccc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.53
DRD2 P14416 4/20 0.49
HTR1A P08908 1/20 0.49
HTR2A P28223 1/20 0.49
HTT P42858 1/20 0.49
DRD4 P21917 6/20 0.48
DRD3 P35462 4/20 0.48
MC4R P32245 1/20 0.46
LMNA P02545 1/20 0.44
POLB P06746 1/20 0.44
OPRM1 P35372 1/20 0.44
OPRK1 P41145 1/20 0.44
ACHE P22303 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12798134 0.80 SIGMAR1 (0.55) SIGMAR1DRD2HTR1AHTR2AHTT
SCHEMBL13959654 0.79 DRD4 (0.56) SIGMAR1DRD2HTR1AHTR2AHTT
SCHEMBL2395932 0.79 DRD4 (0.67) SIGMAR1DRD2HTR1AHTR2AHTT
SCHEMBL1076822 0.79 SIGMAR1 (0.53) SIGMAR1DRD2HTR1AHTR2AHTT
SCHEMBL8831136 0.77 SIGMAR1 (0.52) SIGMAR1DRD2HTR1AHTR2AHTT
SCHEMBL5242533 0.77 SLC6A4 (0.53) SIGMAR1DRD2HTR1AHTR2AHTT
SCHEMBL6263887 0.77 SIGMAR1 (0.52) SIGMAR1DRD2HTR1AHTR2AHTT
Hydrochloric Acid SCHEMBL23882203 0.76 DRD2 (0.50) SIGMAR1DRD2HTR1AHTR2AHTT
SCHEMBL6585625 0.76 DRD4 (0.63) SIGMAR1DRD2HTR1AHTR2AHTT
SCHEMBL8984029 0.76 SIGMAR1 (0.50) SIGMAR1DRD2HTR1AHTR2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3041841-B1 TRIAZOLOPYRIDINE COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF HOFFMANN LA ROCHE (CH) 2019-06-05 EP disclosed
US-5627169-A Selective antagonists for GABArho receptor THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1997-05-06 US disclosed