SCHEMBL8835145

SCHEMBL8835145

C=C/C=C\CC1CCC(c2ccc(F)cc2)CC1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 8/20 0.37
ESR1 P03372 6/20 0.37
CYP2C9 P11712 3/20 0.37
CYP3A4 P08684 2/20 0.37
GRM2 Q14416 2/20 0.33
CYP2D6 P10635 1/20 0.33
HTR1A P08908 2/20 0.32
DRD2 P14416 2/20 0.32
HTR2A P28223 2/20 0.32
DRD3 P35462 2/20 0.32
ACHE P22303 1/20 0.32
DRD1 P21728 1/20 0.32
DRD5 P21918 1/20 0.32
MAP1LC3B Q9GZQ8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8835367 0.96 ESR2 (0.34) ESR2ESR1CYP2C9CYP3A4GRM2
SCHEMBL8835162 0.85 ESR2 (0.40) ESR2ESR1CYP2C9CYP3A4CYP2D6
SCHEMBL8835460 0.84 CCR2 (0.34) ESR2ESR1CYP2C9CYP3A4HTR2A
SCHEMBL8835194 0.84 HTR2C (0.46) ESR2ESR1CYP2C9CYP3A4GRM2
SCHEMBL11308480 0.83 ESR2 (0.41) ESR2ESR1CYP2C9CYP3A4GRM2
SCHEMBL9479280 0.82 ESR2 (0.40) ESR2ESR1CYP2C9CYP3A4GRM2
SCHEMBL9479291 0.82 ESR2 (0.40) ESR2ESR1CYP2C9CYP3A4GRM2
SCHEMBL9479287 0.82 ESR2 (0.40) ESR2ESR1CYP2C9CYP3A4GRM2
SCHEMBL9479295 0.82 ESR2 (0.40) ESR2ESR1CYP2C9CYP3A4GRM2
SCHEMBL8834906 0.82 CYP2C9 (0.38) ESR2ESR1CYP2C9CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5662830-A Diene derivative CHISSO CORPORATION (JP) 1997-09-02 US disclosed
US-5609791-A Diene derivative CHISSO CORPORATION (JP) 1997-03-11 US disclosed
EP-0563982-B1 Polycyclic diene derivatives CHISSO CORP (JP) 1996-07-17 EP disclosed
US-5449810-A Diene derivative CHISSO CORPORATION (JP) 1995-09-12 US disclosed
EP-0563982-A2 Polycyclic diene derivatives Chisso Corporation (JP) 1993-10-06 EP disclosed