SCHEMBL8835367

SCHEMBL8835367

C=C/C=C\CC1CCC(c2ccc(-c3ccc(F)cc3)cc2)CC1

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 7/20 0.34
ESR1 P03372 6/20 0.34
CYP2C9 P11712 3/20 0.34
PTGS1 P23219 2/20 0.34
PTGS2 P35354 2/20 0.34
CYP3A4 P08684 2/20 0.34
DGAT1 O75907 2/20 0.34
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
GRM2 Q14416 2/20 0.32
CYP2D6 P10635 1/20 0.31
HTR1A P08908 1/20 0.30
DRD2 P14416 1/20 0.30
HTR2A P28223 1/20 0.30
DRD3 P35462 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8835145 0.96 ESR2 (0.37) ESR2ESR1CYP2C9CYP3A4GRM2
SCHEMBL8835096 0.86 ESR2 (0.37) ESR2ESR1CYP2C9PTGS1PTGS2
SCHEMBL11033776 0.85 ESR2 (0.38) ESR2ESR1CYP2C9PTGS1PTGS2
SCHEMBL11033780 0.85 ESR2 (0.38) ESR2ESR1CYP2C9PTGS1PTGS2
SCHEMBL8835533 0.85 HTR2C (0.43) ESR2PTGS2DGAT1GRM2HTR1A
SCHEMBL8835301 0.84 DGAT1 (0.33) ESR2ESR1CYP2C9CYP3A4DGAT1
SCHEMBL9477671 0.84 ESR2 (0.37) ESR2ESR1CYP2C9PTGS1PTGS2
SCHEMBL9477665 0.84 ESR2 (0.37) ESR2ESR1CYP2C9PTGS1PTGS2
SCHEMBL9477680 0.84 ESR2 (0.37) ESR2ESR1CYP2C9PTGS1PTGS2
SCHEMBL9477653 0.84 ESR2 (0.37) ESR2ESR1CYP2C9PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5662830-A Diene derivative CHISSO CORPORATION (JP) 1997-09-02 US disclosed
US-5609791-A Diene derivative CHISSO CORPORATION (JP) 1997-03-11 US disclosed
EP-0563982-B1 Polycyclic diene derivatives CHISSO CORP (JP) 1996-07-17 EP disclosed
US-5449810-A Diene derivative CHISSO CORPORATION (JP) 1995-09-12 US disclosed
EP-0563982-A2 Polycyclic diene derivatives Chisso Corporation (JP) 1993-10-06 EP disclosed