SCHEMBL883801

SCHEMBL883801

Cc1cc(C(=O)O)cc2c1OCC[C@H]2NC(=O)c1ccccc1N

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 1/20 0.42
KDM4E B2RXH2 4/20 0.41
ALDH1A1 P00352 4/20 0.41
HSD17B2 P37059 1/20 0.38
HSD17B10 Q99714 2/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
CASP3 P42574 1/20 0.37
SENP8 Q96LD8 1/20 0.37
SENP7 Q9BQF6 1/20 0.37
SENP6 Q9GZR1 1/20 0.37
BRD4 O60885 2/20 0.37
CREBBP Q92793 2/20 0.37
TAS1R3 Q7RTX0 3/20 0.36
TAS1R1 Q7RTX1 3/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
HPGD P15428 1/20 0.36
MAPK1 P28482 1/20 0.35
TAS1R2 Q8TE23 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13190098 0.88 ALDH1A1 (0.47) ALDH1A1NPC1RAB9ATAS1R3TAS1R1
SCHEMBL883780 0.78 ALDH1A1 (0.45) ALDH1A1NPC1RAB9ATAS1R3TAS1R1
SCHEMBL13190008 0.78 ALDH1A1 (0.45) ALDH1A1NPC1RAB9ATAS1R3TAS1R1
SCHEMBL786085 0.75 ALDH1A1 (0.47) ALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL785920 0.75 ALDH1A1 (0.47) ALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL784976 0.69 ALDH1A1 (0.49) ALDH1A1BRD4CREBBPTAS1R3TAS1R1
SCHEMBL484844 0.69 ALDH1A1 (0.49) ALDH1A1BRD4CREBBPTAS1R3TAS1R1
SCHEMBL883818 0.69 ALDH1A1 (0.52) ALDH1A1NPC1RAB9ATAS1R3TAS1R1
SCHEMBL784603 0.68 ALDH1A1 (0.50) ALDH1A1HSD17B2BRD4CREBBPTAS1R3
SCHEMBL784602 0.68 ALDH1A1 (0.50) ALDH1A1HSD17B2BRD4CREBBPTAS1R3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO disclosed