SCHEMBL8838337

SCHEMBL8838337

CC(=O)OCc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.53
ALDH1A1 P00352 2/20 0.48
CES2 O00748 1/20 0.44
TACR1 P25103 8/20 0.44
MAPT P10636 2/20 0.44
CYP3A4 P08684 2/20 0.44
CYP1A2 P05177 2/20 0.44
CYP2C19 P33261 2/20 0.44
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
LMNA P02545 1/20 0.44
TP53 P04637 1/20 0.44
POLB P06746 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
NFKB1 P19838 1/20 0.44
APEX1 P27695 1/20 0.44
THPO P40225 1/20 0.44
BLM P54132 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27799870 0.91 IDO1 (0.44) IDO1ALDH1A1TACR1MAPTCYP3A4
SCHEMBL14255479 0.90 FFAR4 (0.44) IDO1ALDH1A1TACR1MAPTCYP3A4
SCHEMBL27734414 0.89 IDO1 (0.46) IDO1ALDH1A1TACR1MAPTCYP3A4
SCHEMBL27734452 0.83 P2RX1 (0.42) IDO1ALDH1A1MAPTMEN1LMNA
SCHEMBL28778785 0.83 MRGPRX4 (0.38) IDO1ALDH1A1TACR1MAPTCYP3A4
SCHEMBL13292600 0.83 IDO1 (0.47) IDO1ALDH1A1CES2TACR1MAPT
SCHEMBL2660451 0.83 PRKCA (0.63) IDO1ALDH1A1MAPTPRKCAPRKCD
SCHEMBL27800047 0.82 ALDH1A1 (0.41) IDO1ALDH1A1TACR1MAPTCYP3A4
SCHEMBL8838335 0.82 IDO1 (0.50) IDO1ALDH1A1CES2TACR1MAPT
SCHEMBL5663864 0.82 TACR1 (0.42) IDO1CES2TACR1CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7345040-B2 Reverse-turn mimetics and compositions and methods relating thereto MYRIAD GENETICS, INC. (US) 2008-03-18 US disclosed
US-5696267-A ANTIHISTAMINES; ANTIINFLAMMATORY AGENTS; GASTROINTESTINAL DISORDERS SCHERING CORPORATION (US) 1997-12-09 US disclosed