SCHEMBL8840588

SCHEMBL8840588

CCCCOc1ccc(-c2ccc(N(c3ccnc(COC)c3OC)C3CCCCC3)cc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 10/20 0.38
CYP3A4 P08684 5/20 0.38
CYP19A1 P11511 8/20 0.35
CYP2C9 P11712 8/20 0.35
CYP2C19 P33261 8/20 0.35
CYP1A2 P05177 6/20 0.35
HTR2A P28223 1/20 0.34
TRPM8 Q7Z2W7 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
TSHR P16473 1/20 0.32
KCNH2 Q12809 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8840512 0.82 KCNA3 (0.38) CYP3A4TRPM8MEN1KMT2A
SCHEMBL9040850 0.81 NPC1 (0.42) CYP2D6CYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL8840520 0.76 NPC1 (0.41) CYP2D6CYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL9033574 0.75 NPC1 (0.42) CYP2D6CYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL9023787 0.75 BDKRB2 (0.35) TRPM8
SCHEMBL9034144 0.69 NPC1 (0.42) CYP2D6CYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL8840544 0.67 MEN1 (0.36) CYP2D6CYP19A1CYP2C9CYP2C19CYP1A2
SCHEMBL9033513 0.67 KCNA3 (0.41) CYP3A4TRPM8MEN1KMT2AKCNH2
SCHEMBL8463989 0.66 TSHR (0.44) CYP2D6CYP3A4CYP2C9CYP2C19CYP1A2
Hydrochloric Acid SCHEMBL8704982 0.66 KCNA3 (0.40) CYP3A4TRPM8MEN1KMT2AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5650417-A Substituted pyridines, their preparation, and their use as pesticides and fungicides HOECHST SCHERING AGREVO GMBH (DE) 1997-07-22 US disclosed
EP-0719255-A1 SUBSTITUTED PYRIDINES, PROCESS FOR PRODUCING THEM AND THEIR USE AS PESTICIDES AND FUNGICIDES Hoechst Schering AgrEvo GmbH (DE) 1996-07-03 EP disclosed
WO-1995007890-A1 SUBSTITUTED PYRIDINES, PROCESS FOR PRODUCING THEM AND THEIR USE AS PESTICIDES AND FUNGICIDES HOECHST SCHERING AGREVO GMBH (DE) 1995-03-23 WO disclosed