SCHEMBL8842380

SCHEMBL8842380

Brc1cccc(Nc2c[nH]nn2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 2/20 0.43
ABCB1 P08183 1/20 0.43
ABCC1 P33527 1/20 0.43
RAPGEF4 Q8WZA2 1/20 0.42
EGFR P00533 9/20 0.42
IDO1 P14902 1/20 0.41
HTR1A P08908 1/20 0.41
HTR1D P28221 1/20 0.41
HTR1B P28222 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
HTR7 P34969 1/20 0.41
HTR2B P41595 1/20 0.41
HTR5A P47898 1/20 0.41
HTR6 P50406 1/20 0.41
AURKA O14965 1/20 0.41
AURKB Q96GD4 1/20 0.41
INCENP Q9NQS7 1/20 0.41
NCOA1 Q15788 1/20 0.41
NCOA3 Q9Y6Q9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29699515 0.82 MEN1 (0.37) ABCG2ABCB1ABCC1FBP1KDM4E
SCHEMBL23457500 0.82 MEN1 (0.37) ABCG2ABCB1ABCC1FBP1KDM4E
SCHEMBL15831504 0.80 MAPT (0.43) RAPGEF4EGFRKDM4ECDK1MAPT
SCHEMBL3957483 0.80 NPSR1 (0.50) EGFRERBB2ABL1CYP1A2CYP3A4
SCHEMBL828555 0.78 MEN1 (0.48) ABCG2HTR2BAURKAKDM4ECYP1A2
SCHEMBL16881732 0.75 EGFR (0.46) ABCG2ABCB1ABCC1RAPGEF4EGFR
SCHEMBL8842950 0.73 EGFR (0.44) ABCG2ABCB1ABCC1RAPGEF4EGFR
SCHEMBL1687027 0.73 RAPGEF4 (0.61) ABCG2RAPGEF4EGFRIDO1HTR1A
SCHEMBL29961149 0.73 RAPGEF4 (0.61) ABCG2RAPGEF4EGFRIDO1HTR1A
SCHEMBL29961547 0.73 RAPGEF4 (0.61) ABCG2RAPGEF4EGFRIDO1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5679683-A USEFUL FOR TREATING CANCER, ARTHRITIS, PSORIASIS, VASCULAR RESTENOSIS AND ANGIOGENESIS WARNER-LAMBERT COMPANY (US) 1997-10-21 US disclosed