SCHEMBL828555

SCHEMBL828555

c1ccc(Nc2c[nH]nn2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 6/20 0.48
KMT2A Q03164 6/20 0.48
MAPT P10636 5/20 0.48
RAB9A P51151 3/20 0.48
TDP1 Q9NUW8 2/20 0.48
KDM4E B2RXH2 1/20 0.48
ALPG P10696 1/20 0.48
ALDH1A1 P00352 4/20 0.46
LMNA P02545 1/20 0.46
HSD17B10 Q99714 3/20 0.44
TSHR P16473 2/20 0.44
GAA P10253 2/20 0.44
TP53 P04637 1/20 0.44
MAPK1 P28482 2/20 0.42
ALOX15 P16050 1/20 0.42
ALOX12 P18054 1/20 0.42
PTGS1 P23219 1/20 0.42
SLC6A2 P23975 1/20 0.42
PTGS2 P35354 1/20 0.42
HTR2B P41595 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27512047 0.82 ALDH1A1 (0.48) MEN1KMT2AMAPTRAB9ATDP1
SCHEMBL15831504 0.82 MAPT (0.43) MEN1KMT2AMAPTRAB9AKDM4E
SCHEMBL4149136 0.80 MAPK10 (0.49) MEN1KMT2AMAPTRAB9ATDP1
SCHEMBL7049484 0.80 HAO1 (0.49) MEN1KMT2AMAPTRAB9AALDH1A1
SCHEMBL3957483 0.78 NPSR1 (0.50) MEN1KMT2AMAPTRAB9AMAPK1
SCHEMBL8842380 0.78 ABCG2 (0.43) MAPTKDM4ETSHRMAPK1HTR2B
SCHEMBL11337052 0.76 KMT2A (0.53) MEN1KMT2ARAB9ATDP1KDM4E
SCHEMBL10912483 0.74 NPC1 (0.58) MEN1KMT2ARAB9ALMNATSHR
SCHEMBL27672131 0.73 CA1 (0.56) CDK2CDK1ROCK1
SCHEMBL4163888 0.73 KMT2A (0.45) MEN1KMT2AMAPTRAB9ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 187 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4363043-B1 COMPOSITIONS FOR USE IN METHODS FOR INCREASING CANCER CELL SENSITIVITY TO ALTERNATING ELECTRIC FIELDS NOVOCURE GMBH (CH) 2026-04-22 EP claimed
US-12594421-B2 Compositions and methods for increasing cancer cell sensitivity to alternating electric fields NOVOCURE GMBH (CH) 2026-04-07 US claimed
US-20250339680-A1 COMPOSITIONS AND METHODS FOR INCREASING CANCER CELL SENSITIVITY TO ALTERNATING ELECTRIC FIELDS NOVOCURE GMBH (CH) 2025-11-06 US claimed
US-20240316012-A1 METHODS FOR TREATING LYMPHOMA NORTHWESTERN UNIVERSITY (US) 2024-09-26 US claimed
US-20240219403-A1 METHODS FOR INHIBITING KRAS ONCOPROTEIN THROUGH ENHANCED GTPASE ACTIVITY NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2024-07-04 US claimed
EP-4363043-A1 COMPOSITIONS AND METHODS FOR INCREASING CANCER CELL SENSITIVITY TO ALTERNATING ELECTRIC FIELDS Novocure GmbH (CH) 2024-05-08 EP claimed
CN-117580614-A Compositions and methods for increasing sensitivity of cancer cells to alternating electric fields 诺沃库勒有限责任公司 2024-02-20 CN claimed
CN-116390760-A Compositions and methods for increasing sensitivity of cancer cells to alternating electric fields 诺沃库勒有限责任公司 2023-07-04 CN claimed
EP-4188380-A1 COMPOSITIONS AND METHODS FOR INCREASING CANCER CELL SENSITIVITY TO ALTERNATING ELECTRIC FIELDS Novocure GmbH (CH) 2023-06-07 EP claimed
US-20230001193-A1 COMPOSITIONS AND METHODS FOR INCREASING CANCER CELL SENSITIVITY TO ALTERNATING ELECTRIC FIELDS BIOPHARMA CREDIT PLC (GB) 2023-01-05 US claimed
WO-2023275649-A1 COMPOSITIONS AND METHODS FOR INCREASING CANCER CELL SENSITIVITY TO ALTERNATING ELECTRIC FIELDS NOVOCURE GMBH (CH) 2023-01-05 WO claimed
WO-2022217073-A1 METHODS FOR INHIBITING KRAS ONCOPROTEIN THROUGH ENHANCED GTPASE ACTIVITY MEMORIAL SLOAN-KETTERING CANCER CENTER (US) 2022-10-13 WO claimed
CN-114938810-A Thifluzamide and azoxystrobin-containing bactericidal composition suitable for unmanned aerial defense 赤天化科技集团有限公司 2022-08-26 CN claimed
WO-2022093770-A1 COMBINATION THERAPY WITH PI3K-AKT-MTOR INHIBITORS AND FERROPTOSIS INDUCING AGENTS TO TREAT CANCER MEMORIAL SLOAN KETTERING CANCER CENTER (US) 2022-05-05 WO claimed
US-20220096818-A1 Compositions And Methods For Increasing Cancer Cell Sensitivity To Alternating Electric Fields BIOPHARMA CREDIT PLC (GB) 2022-03-31 US claimed
WO-2022029628-A1 COMPOSITIONS AND METHODS FOR INCREASING CANCER CELL SENSITIVITY TO ALTERNATING ELECTRIC FIELDS NOVOCURE GMBH (CH) 2022-02-10 WO claimed
EP-2035436-B1 FUSED THIAZOLE DERIVATIVES AS KINASE INHIBITORS UCB PHARMA SA (BE) 2011-05-25 EP claimed
WO-2006099957-A1 INSECTICIDAL AND ACARICIDAL ANILINOTRIAZOLES BAYER CROPSCIENCE AG (DE) 2006-09-28 WO claimed
EP-0073931-B1 ANILINO-1,2,3-TRIAZOLE DERIVATIVES, MEDICAMENTS CONTAINING THEM, PROCESS FOR PREPARING THEM, AND THEIR USE BOEHRINGER INGELHEIM KG (DE) 1985-02-13 EP claimed
EP-4729067-A2 ELECTRODE ASSEMBLY FOR APPLYING TUMOR TREATING FIELDS WITH A SHEET OF ANISOTROPIC MATERIAL Novocure GmbH (CH) 2026-04-22 EP disclosed
EP-4363043-B1 COMPOSITIONS FOR USE IN METHODS FOR INCREASING CANCER CELL SENSITIVITY TO ALTERNATING ELECTRIC FIELDS NOVOCURE GMBH (CH) 2026-04-22 EP disclosed
US-12594421-B2 Compositions and methods for increasing cancer cell sensitivity to alternating electric fields NOVOCURE GMBH (CH) 2026-04-07 US disclosed
US-20250339680-A1 COMPOSITIONS AND METHODS FOR INCREASING CANCER CELL SENSITIVITY TO ALTERNATING ELECTRIC FIELDS NOVOCURE GMBH (CH) 2025-11-06 US disclosed
US-12415844-B2 BCMA specific VCAR compositions and methods for use POSEIDA THERAPEUTICS, INC. (US) 2025-09-16 US disclosed
US-12383738-B2 Compositions and methods for increasing cancer cell sensitivity to alternating electric fields NOVOCURE GMBH (CH) 2025-08-12 US disclosed
US-20250171518-A1 METHODS FOR PREPARING CELLS FOR ADOPTIVE T CELL THERAPY CITY OF HOPE 2025-05-29 US disclosed
US-20250025473-A1 CELL IMPERMEABLE KINASE INHIBITORS TO TREAT SARS-COV-2 AND/OR HSV VIRAL INFECTIONS ALBERT EINSTEIN COLLEGE MEDICINE (US) 2025-01-23 US disclosed
US-20250001166-A1 COMPOSITIONS AND METHODS FOR INCREASING CANCER CELL SENSITIVITY TO ALTERNATING ELECTRIC FIELDS NOVOCURE GMBH (CH) 2025-01-02 US disclosed
CN-119119296-A Allogeneic cell compositions and methods of use 波赛达治疗公司 2024-12-13 CN disclosed
CN-118878697-A VCAR compositions and methods of use 波赛达治疗公司 2024-11-01 CN disclosed
US-20240316012-A1 METHODS FOR TREATING LYMPHOMA NORTHWESTERN UNIVERSITY (US) 2024-09-26 US disclosed
CN-113383018-B Allogeneic cell compositions and methods of use 波赛达治疗公司 2024-09-10 CN disclosed
EP-4413038-A1 PD-L1 BINDING AFFIMERS Avacta Life Sciences Limited (GB) 2024-08-14 EP disclosed
EP-4412711-A1 SERUM HALF-LIFE EXTENDED PD-L1 BINDING POLYPEPTIDES Avacta Life Sciences Limited (GB) 2024-08-14 EP disclosed
US-20240219403-A1 METHODS FOR INHIBITING KRAS ONCOPROTEIN THROUGH ENHANCED GTPASE ACTIVITY NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2024-07-04 US disclosed
US-20240207292-A1 BORONIC ACID COMPOUNDS, COMPOSITIONS AND METHODS TRUSTEES OF TUFTS COLLEGE 2024-06-27 US disclosed
CN-112218885-B VCAR compositions and methods of use 波赛达治疗公司 2024-06-18 CN disclosed
US-12005253-B2 Compositions and methods for increasing cancer cell sensitivity to alternating electric fields NOVOCURE GMBH (CH) 2024-06-11 US disclosed
US-20240166759-A1 COMBINATIONS COMPRISING ANTI-TM4SF1 ANTIBODIES AND IMMUNOTHERAPEUTIC AGENTS AND METHODS OF USING THE SAME ANGIEX, INC. 2024-05-23 US disclosed
EP-4363043-A1 COMPOSITIONS AND METHODS FOR INCREASING CANCER CELL SENSITIVITY TO ALTERNATING ELECTRIC FIELDS Novocure GmbH (CH) 2024-05-08 EP disclosed
EP-4344414-A1 ELECTRODE ASSEMBLY FOR APPLYING TUMOR TREATING FIELDS (TTFIELDS) WITH A SHEET OF ANISOTROPIC MATERIAL Novocure GmbH (CH) 2024-04-03 EP disclosed
CN-117580614-A Compositions and methods for increasing sensitivity of cancer cells to alternating electric fields 诺沃库勒有限责任公司 2024-02-20 CN disclosed
EP-4313033-A1 BORONIC ACID COMPOUNDS, COMPOSITIONS AND METHODS TRUSTEES OF TUFTS COLLEGE (US) 2024-02-07 EP disclosed
EP-4313144-A1 COMBINATIONS COMPRISING ANTI-TM4SF1 ANTIBODIES AND IMMUNOTHERAPEUTIC AGENTS AND METHODS OF USING THE SAME Angiex, Inc. (US) 2024-02-07 EP disclosed
CN-117425476-A Boric acid compounds, compositions and methods 塔夫茨大学的受托人 2024-01-19 CN disclosed
CN-117355333-A Combination comprising anti-TM 4SF1 antibody and immunotherapeutic agent and method of use thereof 安吉克公司 2024-01-05 CN disclosed
WO-2023218243-A1 LAG-3/PD-L1 BINDING FUSION PROTEINS AVACTA LIFE SCIENCES LIMITED (GB) 2023-11-16 WO disclosed
EP-4262878-A1 FAP-ACTIVATED RADIOTHERANOSTICS, AND USES RELATED THERETO TRUSTEES OF TUFTS COLLEGE (US) 2023-10-25 EP disclosed
US-20230330275-A1 FAP-TARGETED RADIOPHARMACEUTICALS AND IMAGING AGENTS, AND USES RELATED THERETO TRUSTEES OF TUFTS COLLEGE 2023-10-19 US disclosed
US-11707539-B2 FAP-targeted radiopharmaceuticals and imaging agents, and uses related thereto TRUSTEES OF TUFTS COLLEGE (US) 2023-07-25 US disclosed
CN-116390760-A Compositions and methods for increasing sensitivity of cancer cells to alternating electric fields 诺沃库勒有限责任公司 2023-07-04 CN disclosed
EP-4188380-A1 COMPOSITIONS AND METHODS FOR INCREASING CANCER CELL SENSITIVITY TO ALTERNATING ELECTRIC FIELDS Novocure GmbH (CH) 2023-06-07 EP disclosed
EP-4185586-A1 NOVEL COMPOUNDS AS HISTONE DEACETYLASE 6 INHIBITOR, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME Chong Kun Dang Pharmaceutical Corp. (KR) 2023-05-31 EP disclosed
CN-116157398-A 2- (4- ((5- (benzo [ b ] thiophen-3-yl) -1H-tetrazol-1-yl) methyl) phenyl) -5- (difluoromethyl) -1,3, 4-oxadiazole derivatives and similar compounds as selective inhibitors of histone deacetylase 6 (HDAC 6) for the treatment of, for example, peripheral neuropathy 意大发马克股份公司 2023-05-23 CN disclosed
WO-2023086547-A1 CELL IMPERMEABLE KINASE INHIBITORS TO TREAT SARS-COV-2 AND/OR HSV VIRAL INFECTIONS ALBERT EINSTEIN COLLEGE OF MEDICINE (US) 2023-05-19 WO disclosed
US-20230149295-A1 INFLAMMATORY BOWEL DISEASE STEM CELLS, AGENTS WHICH TARGET IBD STEM CELLS, AND USES RELATED THERETO UNIVERSITY OF HOUSTON SYSTEM (US) 2023-05-18 US disclosed
CN-116133658-A Novel compounds as inhibitors of histone deacetylase 6 and pharmaceutical compositions comprising the same 株式会社 钟根堂 2023-05-16 CN disclosed
US-20230121433-A1 CHIMERIC STIMULATORY RECEPTORS AND METHODS OF USE IN T CELL ACTIVATION AND DIFFERENTIATION POSEIDA THERAPEUTICS, INC. 2023-04-20 US disclosed
WO-2023057946-A1 SERUM HALF-LIFE EXTENDED PD-L1 BINDING POLYPEPTIDES AVACTA LIFE SCIENCES LIMITED (GB) 2023-04-13 WO disclosed
WO-2023057567-A1 PD-L1 BINDING AFFIMERS AVACTA LIFE SCIENCES LIMITED (GB) 2023-04-13 WO disclosed
WO-2023012707-A1 ELECTRODE ASSEMBLY FOR APPLYING TUMOR TREATING FIELDS (TTFIELDS) WITH A SHEET OF ANISOTROPIC MATERIAL NOVOCURE GMBH (CH) 2023-02-09 WO disclosed
US-20230037806-A1 Electrode Assembly for Applying Tumor Treating Fields (TTFields) with a Sheet of Anisotropic Material NOVOCURE GMBH (CH) 2023-02-09 US disclosed
US-20230039099-A1 AKT INHIBITORS FOR ENHANCING CHIMERIC T CELL PERSISTENCE H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. 2023-02-09 US disclosed
EP-4126053-A1 FAP-TARGETED RADIOPHARMACEUTICALS AND IMAGING AGENTS, AND USES RELATED THERETO TRUSTEES OF TUFTS COLLEGE (US) 2023-02-08 EP disclosed
CN-115697413-A Radiopharmaceuticals and imaging agents targeting FAP and uses related thereto 塔夫茨大学信托人 2023-02-03 CN disclosed
EP-4121111-A1 METHODS AND COMPOSITIONS FOR TREATING INFLAMMATORY AND FIBROTIC PULMONARY DISORDERS University of Houston System (US) 2023-01-25 EP disclosed
EP-4118107-A1 CHIMERIC STIMULATORY RECEPTORS AND METHODS OF USE IN T CELL ACTIVATION AND DIFFERENTIATION Poseida Therapeutics, Inc. (US) 2023-01-18 EP disclosed
EP-4117718-A1 INFLAMMATORY BOWEL DISEASE STEM CELLS, AGENTS WHICH TARGET IBD STEM CELLS, AND USES RELATED THERETO University of Houston System (US) 2023-01-18 EP disclosed
US-20230001193-A1 COMPOSITIONS AND METHODS FOR INCREASING CANCER CELL SENSITIVITY TO ALTERNATING ELECTRIC FIELDS BIOPHARMA CREDIT PLC (GB) 2023-01-05 US disclosed
WO-2023275649-A1 COMPOSITIONS AND METHODS FOR INCREASING CANCER CELL SENSITIVITY TO ALTERNATING ELECTRIC FIELDS NOVOCURE GMBH (CH) 2023-01-05 WO disclosed
US-20220395575-A1 COMBINATION THERAPY WITH PROTEIN KINASE B ACTIVATION INHIBITOR TO TREAT CANCER H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. 2022-12-15 US disclosed
US-20220389077-A1 ALLOGENEIC CELL COMPOSITIONS AND METHODS OF USE POSEIDA THERAPEUTICS, INC. 2022-12-08 US disclosed
US-20220372491-A1 TREATMENT OF RENAL CYSTIC DISEASE MONASH UNIVERSITY (AU) 2022-11-24 US disclosed
US-20220370647-A1 FAP-TARGETED RADIOPHARMACEUTICALS AND IMAGING AGENTS, AND USES RELATED THERETO TRUSTEES OF TUFTS COLLEGE 2022-11-24 US disclosed
WO-2022234003-A1 CD33 BINDING POLYPEPTIDES WITH STEFIN A PROTEIN AVACTA LIFE SCIENCES LIMITED (GB) 2022-11-10 WO disclosed
WO-2022217073-A1 METHODS FOR INHIBITING KRAS ONCOPROTEIN THROUGH ENHANCED GTPASE ACTIVITY MEMORIAL SLOAN-KETTERING CANCER CENTER (US) 2022-10-13 WO disclosed
CN-115175686-A AKT inhibitors for enhancing persistence of chimeric T cells H·李·莫菲特癌症中心研究所公司 2022-10-11 CN disclosed
WO-2022204368-A1 BORONIC ACID COMPOUNDS, COMPOSITIONS AND METHODS TRUSTEES OF TUFTS COLLEGE (US) 2022-09-29 WO disclosed
WO-2022204565-A1 COMBINATIONS COMPRISING ANTI-TM4SF1 ANTIBODIES AND IMMUNOTHERAPEUTIC AGENTS AND METHODS OF USING THE SAME ANGIEX, INC. (US) 2022-09-29 WO disclosed
EP-4061383-A1 AKT INHIBITORS FOR ENHANCING CHIMERIC T CELL PERSISTENCE H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE INC. (US) 2022-09-28 EP disclosed
EP-4051273-A1 TREATMENT OF RENAL CYSTIC DISEASE Monash University (AU) 2022-09-07 EP disclosed
CN-114938810-A Thifluzamide and azoxystrobin-containing bactericidal composition suitable for unmanned aerial defense 赤天化科技集团有限公司 2022-08-26 CN disclosed
US-20220259673-A1 METHODS FOR IDENTIFYING AND TREATING HIGH-PLASTICITY CELL STATE DRIVING TUMOR PROGRESSION IN LUNG CANCER MEMORIAL SLOAN KETTERING CANCER CENTER (US) 2022-08-18 US disclosed
US-20220211883-A1 FAP-ACTIVATED RADIOTHERANOSTICS AND USES RELATED THERETO TRUSTEES OF TUFTS COLLEGE 2022-07-07 US disclosed
WO-2022133288-A1 FAP-ACTIVATED RADIOTHERANOSTICS, AND USES RELATED THERETO TRUSTEES OF TUFTS COLLEGE (US) 2022-06-23 WO disclosed
WO-2022093770-A1 COMBINATION THERAPY WITH PI3K-AKT-MTOR INHIBITORS AND FERROPTOSIS INDUCING AGENTS TO TREAT CANCER MEMORIAL SLOAN KETTERING CANCER CENTER (US) 2022-05-05 WO disclosed
US-20220096818-A1 Compositions And Methods For Increasing Cancer Cell Sensitivity To Alternating Electric Fields BIOPHARMA CREDIT PLC (GB) 2022-03-31 US disclosed
WO-2022029628-A1 COMPOSITIONS AND METHODS FOR INCREASING CANCER CELL SENSITIVITY TO ALTERNATING ELECTRIC FIELDS NOVOCURE GMBH (CH) 2022-02-10 WO disclosed
US-20210401987-A1 METHODS AND COMPOSITIONS FOR TREATING INFLAMMATORY AND FIBROTIC PULMONARY DISORDERS UNIVERSITY OF HOUSTON SYSTEM (US) 2021-12-30 US disclosed
WO-2021195198-A1 FAP-TARGETED RADIOPHARMACEUTICALS AND IMAGING AGENTS, AND USES RELATED THERETO TRUSTEES OF TUFTS COLLEGE (US) 2021-09-30 WO disclosed
WO-2021188849-A1 METHODS AND COMPOSITIONS FOR TREATING INFLAMMATORY AND FIBROTIC PULMONARY DISORDERS UNIVERSITY OF HOUSTON SYSTEM (US) 2021-09-23 WO disclosed
WO-2021183474-A1 INFLAMMATORY BOWEL DISEASE STEM CELLS, AGENTS WHICH TARGET IBD STEM CELLS, AND USES RELATED THERETO UNIVERSITY OF HOUSTON SYSTEM (US) 2021-09-16 WO disclosed
WO-2021183795-A1 CHIMERIC STIMULATORY RECEPTORS AND METHODS OF USE IN T CELL ACTIVATION AND DIFFERENTIATION POSEIDA THERAPEUTICS, INC. (US) 2021-09-16 WO disclosed
CN-113383018-A Allogeneic cell compositions and methods of use 波赛达治疗公司 2021-09-10 CN disclosed
EP-3847197-A1 ALLOGENEIC CELL COMPOSITIONS AND METHODS OF USE Poseida Therapeutics, Inc. (US) 2021-07-14 EP disclosed
US-20210163599-A1 PD-L1 BINDING AFFIMERS, AND USES RELATED THERETO AVACTA LIFE SCIENCES LIMITED (GB) 2021-06-03 US disclosed
WO-2021102038-A1 AKT INHIBITORS FOR ENHANCING CHIMERIC T CELL PERSISTENCE H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE INC. (US) 2021-05-27 WO disclosed
WO-2021097401-A1 COMBINATION THERAPY WITH PROTEIN KINASE B ACTIVATION INHIBITOR TO TREAT CANCER H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. (US) 2021-05-20 WO disclosed
US-20210139557-A1 VCAR COMPOSITIONS AND METHODS FOR USE POSEIDA THERAPEUTICS, INC. 2021-05-13 US disclosed
WO-2021081580-A1 TREATMENT OF RENAL CYSTIC DISEASE MONASH UNIVERSITY (AU) 2021-05-06 WO disclosed
US-20210130845-A1 COMPOSITIONS AND METHODS FOR CHIMERIC LIGAND RECEPTOR (CLR)-MEDIATED CONDITIONAL GENE EXPRESSION POSEIDA THERAPEUTICS, INC. 2021-05-06 US disclosed
WO-2021074695-A1 PD-L1 INHIBITOR - TGFβ INHIBITOR BISPECIFIC DRUG MOIETIES. AVACTA LIFE SCIENCES LIMITED (GB) 2021-04-22 WO disclosed
US-20210107993-A1 CARTYRIN COMPOSITIONS AND METHODS FOR USE POSEIDA THERAPEUTICS, INC. 2021-04-15 US disclosed
US-20210102165-A1 METHODS FOR PREPARING CELLS FOR ADOPTIVE T CELL THERAPY NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2021-04-08 US disclosed
CN-112601583-A CARTyrin compositions and methods of use 波赛达治疗公司 2021-04-02 CN disclosed
EP-3774868-A1 PD-L1 BINDING AFFIMERS, AND USES RELATED THERETO Avacta Life Sciences Limited (GB) 2021-02-17 EP disclosed
EP-3762106-A1 CARTYRIN COMPOSITIONS AND METHODS FOR USE Poseida Therapeutics, Inc. (US) 2021-01-13 EP disclosed
CN-112218885-A VCAR compositions and methods of use 波赛达治疗公司 2021-01-12 CN disclosed
WO-2019173636-A9 CARTYRIN COMPOSITIONS AND METHODS FOR USE POSEIDA THERAPEUTICS, INC. (US) 2020-11-05 WO disclosed
EP-3728305-A1 VCAR COMPOSITIONS AND METHODS FOR USE Poseida Therapeutics, Inc. (US) 2020-10-28 EP disclosed
CN-111727256-A Compositions and methods for Chimeric Ligand Receptor (CLR) -mediated conditional gene expression 波赛达治疗公司 2020-09-29 CN disclosed
EP-3679145-A2 COMPOSITIONS AND METHODS FOR CHIMERIC LIGAND RECEPTOR (CLR)-MEDIATED CONDITIONAL GENE EXPRESSION Poseida Therapeutics, Inc. (US) 2020-07-15 EP disclosed
WO-2019197583-A1 PD-L1 BINDING AFFIMERS, AND USES RELATED THERETO AVACTA LIFE SCIENCES LIMITED (GB) 2019-10-17 WO disclosed
WO-2019173636-A1 CARTYRIN COMPOSITIONS AND METHODS FOR USE POSEIDA THERAPEUTICS, INC. (US) 2019-09-12 WO disclosed
WO-2019104065-A1 ANTI-AGING METHODS AND COMPOSITIONS TURRINII PHARMACEUTICAL, LLC (US) 2019-05-31 WO disclosed
WO-2019051424-A2 COMPOSITIONS AND METHODS FOR CHIMERIC LIGAND RECEPTOR (CLR)-MEDIATED CONDITIONAL GENE EXPRESSION POSEIDA THERAPEUTICS, INC. (US) 2019-03-14 WO disclosed
EP-2683714-B1 II (PI)-CONJUGATED FLUOROIONOPHORES AND METHOD FOR DETERMINING AN ALKALI ION UNIV POTSDAM (DE) 2019-01-09 EP disclosed
US-20180320133-A1 METHODS FOR PREPARING CELLS FOR ADOPTIVE T CELL THERAPY NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2018-11-08 US disclosed
EP-3370743-A1 METHODS FOR PREPARING CELLS FOR ADOPTIVE T CELL THERAPY City of Hope (US) 2018-09-12 EP disclosed
EP-2782922-B1 ANTIBACTERIAL TYLOSIN DERIVATIVES AND METHODS FOR THEIR PREPARATION BAYER IP GMBH (DE) 2017-12-20 EP disclosed
WO-2017079528-A9 METHODS FOR PREPARING CELLS FOR ADOPTIVE T CELL THERAPY CITY OF HOPE (US) 2017-06-15 WO disclosed
WO-2017079528-A1 METHODS FOR PREPARING CELLS FOR ADOPTIVE T CELL THERAPY CITY OF HOPE (US) 2017-05-11 WO disclosed
US-9593140-B2 Antibacterial tylosin derivatives and methods for their preparation BAYER INTELLECTUAL PROPERTY GMBH (DE) 2017-03-14 US disclosed
US-9499497-B2 Compounds useful as inhibitors of indoleamine 2,3-dioxygenase VERTEX PHARMACEUTICALS INCORPORATED (US) 2016-11-22 US disclosed
US-20150336903-A1 COMPOUNDS USEFUL AS INHIBITORS OF INDOLEAMINE 2,3-DIOXYGENASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2015-11-26 US disclosed
US-9073875-B2 Compounds useful as inhibitors of indoleamine 2,3-dioxygenase VERTEX PHARMACEUTICALS INCORPORATED (US) 2015-07-07 US disclosed
EP-2855698-A2 TARGETING THE GLUTAMINE TO PYRUVATE PATHWAY FOR TREATMENT OF ONCOGENIC KRAS-ASSOCIATED CANCER Dana-Farber Cancer Institute, Inc. (US) 2015-04-08 EP disclosed
CN-104312003-A High-resistance polypropylene sheet Hefei daan printing co ltd 2015-01-28 CN disclosed
CN-104302653-A Antibacterial tylosin derivatives and methods for their preparation BAYER IP GMBH 2015-01-21 CN disclosed
US-20140349954-A1 ANTIBACTERIAL TYLOSIN DERIVATIVES AND METHODS FOR THEIR PREPARATION ELANCO ANIMAL HEALTH GMBH (DE) 2014-11-27 US disclosed
EP-2010516-B1 TRISUBSTITUTED 1,2,4-TRIAZOLES JANSSEN PHARMACEUTICA NV (BE) 2014-07-02 EP disclosed
CN-101472911-B Trisubstituted 1,2,4-triazoles JANSSEN PHARMACEUTICA NV 2014-07-02 CN disclosed
US-20140179699-A1 COMPOUNDS USEFUL AS INHIBITORS OF INDOLEAMINE 2,3-DIOXYGENASE VERTEX PHARMACEUTICALS INCORPORATED 2014-06-26 US disclosed
CN-103666391-A Composite antifreezing solution composition formula QINGDAO CHENXUTONG COMMERCE & TRADE CO LTD 2014-03-26 CN disclosed
US-20130344607-A1 PI-CONJUGATED FLUOROIONOPHORES AND METHOD FOR DETERMINING AN ALKALI ION UNIVERSITAET POTSDAM (DE) 2013-12-26 US disclosed
WO-2013177426-A2 TARGETING THE GLUTAMINE TO PYRUVATE PATHWAY FOR TREATMENT OF ONCOGENIC KRAS-ASSOCIATED CANCER DANA-FARBER CANCER INSTITUTE, INC. (US) 2013-11-28 WO disclosed
CN-103160255-A Motor vehicle antifreeze fluid with good stability QINGDAO WENSHENG AUTOMOBILE COMPONENTS & PARTS CO LTD 2013-06-19 CN disclosed
CN-101489525-B Use of aminophenylbenzotriazole derivatives for protecting human and animal skin and hair from the harmful effects of UV radiation and cosmetic compositions thereof CIBA HOLDING INC 2013-06-19 CN disclosed
US-8242116-B2 Fused thiazole derivatives as kinase inhibitors UCB PHARMA S.A. (BE) 2012-08-14 US disclosed
US-8143419-B2 Trisubstituted 1,2,4-triazoles JANSSEN PHARMACEUTICA N. V. (BE) 2012-03-27 US disclosed
EP-2035436-B1 FUSED THIAZOLE DERIVATIVES AS KINASE INHIBITORS UCB PHARMA SA (BE) 2011-05-25 EP disclosed
EP-1981876-B1 TRIAZOLOANILINOPYRIMIDINE DERIVATIVES FOR USE AS ANTIVIRAL AGENTS ARROW THERAPEUTICS LTD (GB) 2011-05-04 EP disclosed
EP-2207770-A1 1, 2, 3-TRIAZOLE DERIVATIVES FOR USE AS STEAROYL-COA DESATURASE INHIBITORS GlaxoSmithKline LLC (US) 2010-07-21 EP disclosed
US-20100158863-A1 TRIAZOLOANILINOPYRIMIDINE DERIVATIVES FOR USE AS ANTIVIRAL AGENTS ARROW THERAPEUTICS LIMITED (GB) 2010-06-24 US disclosed
US-20100137302-A1 Fused Thiazole Derivatives as Kinase Inhibitors UCB PHARMA S.A. (BE) 2010-06-03 US disclosed
EP-1663211-B1 AMINOTRIAZOLE COMPOUNDS USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2010-01-20 EP disclosed
US-20090253691-A1 TRISUBSTITUTED 1,2,4-TRIAZOLES JANSSEN PHARMACEUTICA N.V. (BE) 2009-10-08 US disclosed
WO-2009122148-A1 FUSED THIOPHENE AND THIAZOLE DERIVATIVES AS PI3K KINASE INHIBITORS UCB PHARMA S.A. (BE) 2009-10-08 WO disclosed
US-7598245-B2 Aminotriazole compounds useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-10-06 US disclosed
CN-101472911-A Trisubstituted 1,2,4-triazoles JANSSEN PHARMACEUTICA NV (BE) 2009-07-01 CN disclosed
WO-2009071888-A1 PYRROLOTHIAZOLES AS PI3-KINASE INHIBITORS UCB PHARMA S.A. (BE) 2009-06-11 WO disclosed
WO-2009071890-A1 TRICYCLIC KINASE INHIBITORS UCB PHARMA S.A. (BE) 2009-06-11 WO disclosed
WO-2009071895-A1 FUSED THIAZOLE AND THIOPHENE DERIVATIVES AS KINASE INHIBITORS UCB PHARMA S.A. (BE) 2009-06-11 WO disclosed
WO-2009060053-A1 1, 2, 3-TRIAZOLE DERIVATIVES FOR USE AS STEAROYL-COA DESATURASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2009-05-14 WO disclosed
EP-2035436-A1 FUSED THIAZOLE DERIVATIVES AS KINASE INHIBITORS UCB Pharma S.A. (BE) 2009-03-18 EP disclosed
CN-101370802-A Triazoloanilinopyrimidine derivatives for use as antiviral agents ARROW THERAPEUTICS LTD (GB) 2009-02-18 CN disclosed
EP-2010516-A1 TRISUBSTITUTED 1,2,4-TRIAZOLES JANSSEN PHARMACEUTICA N.V. (BE) 2009-01-07 EP disclosed
EP-1981876-A1 TRIAZOLOANILINOPYRIMIDINE DERIVATIVES FOR USE AS ANTIVIRAL AGENTS Arrow Therapeutics Limited (GB) 2008-10-22 EP disclosed
US-20080096901-A1 Aminotriazole compounds useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED 2008-04-24 US disclosed
WO-2008001076-A1 FUSED THIAZOLE DERIVATIVES AS KINASE INHIBITORS UCB PHARMA S.A. (BE) 2008-01-03 WO disclosed
WO-2007118903-A1 TRISUBSTITUTED 1,2,4-TRIAZOLES JANSSEN PHARMACEUTICA N.V. (BE) 2007-10-25 WO disclosed
WO-2007080401-A1 TRIAZOLOANILINOPYRIMIDINE DERIVATIVES FOR USE AS ANTIVIRAL AGENTS ARROW THERAPEUTICS LIMITED (GB) 2007-07-19 WO disclosed
US-7226920-B2 Aminotriazole compounds useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INC. (US) 2007-06-05 US disclosed
JP-2006265209-A INSECTICIDAL ANILINOTRIAZOLE COMPOUNDS BAYER CROPSCIENCE AG 2006-10-05 JP disclosed
WO-2006099957-A1 INSECTICIDAL AND ACARICIDAL ANILINOTRIAZOLES BAYER CROPSCIENCE AG (DE) 2006-09-28 WO disclosed
WO-2006099957-A1 INSECTICIDAL AND ACARICIDAL ANILINOTRIAZOLES BAYER CROPSCIENCE AG (DE) 2006-09-28 WO disclosed
US-20050261268-A1 Aminotriazole compounds useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED 2005-11-24 US disclosed
CN-1053660-C Process for preparing indole derivatives containing 1,2,4-triazol-1-yl substituents MERCK SHARP & DOHME (GB) 2000-06-21 CN disclosed
CN-1037843-C Process for preparing indole derivatives containing 1,2, 4-triazol-1-yl substituents MERCK SHARP & DOHME (GB) 1998-03-25 CN disclosed
US-5717104-A Process for preparing indole derivatives containing a 1,2,4-triazol-1-yl substituent MERCK, SHARP & DOHME, LTD. (GB) 1998-02-10 US disclosed
CN-1166486-A Process for preparing indole derivatives containing 1,2,4-triazol-1-yl substituents MERCK SHARP & DOHME (GB) 1997-12-03 CN disclosed
EP-0651748-B1 PROCESS FOR PREPARING INDOLE DERIVATIVES CONTAINING A 1,2,4-TRIAZOL-1-YL SUBSTITUENT MERCK SHARP & DOHME (GB) 1997-10-08 EP disclosed
EP-0679647-B1 Novel antifungal triazole compound and production and use thereof NIHON NOHYAKU CO LTD (JP) 1997-06-04 EP disclosed
US-5629332-A FUNGICIDES NIHON NOHYAKU CO., LTD. (JP) 1997-05-13 US disclosed
US-5567819-A Process for preparing indole derivatives containing a 1,2,4-triazol-1-yl substituent MERCK, SHARP & DOHME, LTD. (GB) 1996-10-22 US disclosed
EP-0679647-A1 Novel antifungal triazole compound and production and use thereof NIHON NOHYAKU CO., LTD. (JP) 1995-11-02 EP disclosed
EP-0651748-A1 PROCESS FOR PREPARING INDOLE DERIVATIVES CONTAINING A 1,2,4-TRIAZOL-1-YL SUBSTITUENT. MERCK SHARP & DOHME (GB) 1995-05-10 EP disclosed
WO-1994002476-A1 PROCESS FOR PREPARING INDOLE DERIVATIVES CONTAINING A 1,2,4-TRIAZOL-1-YL SUBSTITUENT MERCK SHARP & DOHME LIMITED (GB) 1994-02-03 WO disclosed
US-4505912-A SLEEP POTENTIATORS AND BLOOD CIRCULATION ENHANCERS BOEHRINGER INGELHEIM KG (DE) 1985-03-19 US disclosed
EP-0073931-B1 ANILINO-1,2,3-TRIAZOLE DERIVATIVES, MEDICAMENTS CONTAINING THEM, PROCESS FOR PREPARING THEM, AND THEIR USE BOEHRINGER INGELHEIM KG (DE) 1985-02-13 EP disclosed
US-4492699-A NERVOUS SYSTEM DISORDERS LILLY INDUSTRIES LIMITED (GB) 1985-01-08 US disclosed
EP-0040357-B1 PROCESS FOR THE PREPARATION OF V-TRIAZOLYL-(2) PHENOLS BAYER AG (DE) 1984-09-19 EP disclosed
US-4431589-A NEUROLEPTIC AGENTS; TRANQUILIZERS; CENTRAL NERVOUS SYSTEM DISORDERS Lilly House (GB) 1984-02-14 US disclosed
EP-0073931-A1 Anilino-1,2,3-triazole derivatives, medicaments containing them, process for preparing them, and their use BOEHRINGER INGELHEIM KG (DE) 1983-03-16 EP disclosed
EP-0073931-A1 Anilino-1,2,3-triazole derivatives, medicaments containing them, process for preparing them, and their use BOEHRINGER INGELHEIM KG (DE) 1983-03-16 EP disclosed
EP-0054416-A2 Benzodiazepine compounds and their use as pharmaceuticals Lilly Industries Limited (GB) 1982-06-23 EP disclosed
EP-0040357-A1 Process for the preparation of v-triazolyl-(2) phenols BAYER AG (DE) 1981-11-25 EP disclosed
EP-0040357-A1 Process for the preparation of v-triazolyl-(2) phenols BAYER AG (DE) 1981-11-25 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (22 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210401987-A1 METHODS AND COMPOSITIONS FOR TREATING INFLAMMATORY AND FIBROTIC PULMONARY DISORDERS MMP1, MMP8, CCL11 MEN1 4853/4885KMT2A 4026/4885MAPT 3332/4885
US-20100158863-A1 TRIAZOLOANILINOPYRIMIDINE DERIVATIVES FOR USE AS ANTIVIRAL AGENTS SLC28A1, TPMT, ACE MEN1 4286/4885KMT2A 3712/4885MAPT 2681/4885
US-20180320133-A1 METHODS FOR PREPARING CELLS FOR ADOPTIVE T CELL THERAPY CD4, ICOS, CD2 MEN1 3640/4885KMT2A 1396/4885MAPT 2971/4885
US-20230330275-A1 FAP-TARGETED RADIOPHARMACEUTICALS AND IMAGING AGENTS, AND USES RELATED THERETO FAP, APC, FIBP MEN1 1985/4885KMT2A 4040/4885MAPT 1967/4885
US-20250171518-A1 METHODS FOR PREPARING CELLS FOR ADOPTIVE T CELL THERAPY CD4, ICOS, CD2 MEN1 3640/4885KMT2A 1396/4885MAPT 2971/4885
US-20220370647-A1 FAP-TARGETED RADIOPHARMACEUTICALS AND IMAGING AGENTS, AND USES RELATED THERETO FAP, APC, FIBP MEN1 1985/4885KMT2A 4040/4885MAPT 1967/4885
US-11707539-B2 FAP-targeted radiopharmaceuticals and imaging agents, and uses related thereto FAP, APC, FIBP MEN1 1985/4885KMT2A 4040/4885MAPT 1967/4885
US-12594421-B2 Compositions and methods for increasing cancer cell sensitivity to alternating electric fields PTK2, GSK3B, MTOR MEN1 1645/4885KMT2A 2872/4885MAPT 1987/4885
US-20080096901-A1 Aminotriazole compounds useful as inhibitors of protein kinases MAP3K20, MAP3K5, MAP3K1 MEN1 2530/4885KMT2A 508/4885MAPT 599/4885
US-20220211883-A1 FAP-ACTIVATED RADIOTHERANOSTICS AND USES RELATED THERETO FAP, FIBP, FGFR1 MEN1 3078/4885KMT2A 3435/4885MAPT 3059/4885
US-20140349954-A1 ANTIBACTERIAL TYLOSIN DERIVATIVES AND METHODS FOR THEIR PREPARATION MLN, TMSB10, TMSB4X MEN1 3664/4885KMT2A 3403/4885MAPT 2502/4885
US-20230149295-A1 INFLAMMATORY BOWEL DISEASE STEM CELLS, AGENTS WHICH TARGET IBD STEM CELLS, AND USES RELATED THERETO EPCAM, FABP2, TPMT MEN1 4832/4885KMT2A 577/4885MAPT 4173/4885
US-20150336903-A1 COMPOUNDS USEFUL AS INHIBITORS OF INDOLEAMINE 2,3-DIOXYGENASE IDO1, IDO2, INMT MEN1 954/4885KMT2A 518/4885MAPT 2788/4885
US-20100137302-A1 Fused Thiazole Derivatives as Kinase Inhibitors PI4KA, PDPK1, PIK3CA MEN1 1461/4885KMT2A 2966/4885MAPT 955/4885
US-20130344607-A1 PI-CONJUGATED FLUOROIONOPHORES AND METHOD FOR DETERMINING AN ALKALI ION SLCO2A1, SLCO2B1, SLCO4C1 MEN1 1475/4885KMT2A 1767/4885MAPT 3263/4885
US-20250025473-A1 CELL IMPERMEABLE KINASE INHIBITORS TO TREAT SARS-COV-2 AND/OR HSV VIRAL INFECTIONS PDPK1, DAPK1, DAPK2 MEN1 2932/4885KMT2A 2700/4885MAPT 900/4885
US-20050261268-A1 Aminotriazole compounds useful as inhibitors of protein kinases MAP3K20, MAP3K5, MAP3K1 MEN1 2530/4885KMT2A 508/4885MAPT 599/4885
US-20240207292-A1 BORONIC ACID COMPOUNDS, COMPOSITIONS AND METHODS BCL6B, BCL6, BTD MEN1 180/4885KMT2A 1084/4885MAPT 1308/4885
US-20140179699-A1 COMPOUNDS USEFUL AS INHIBITORS OF INDOLEAMINE 2,3-DIOXYGENASE IDO1, IDO2, INMT MEN1 954/4885KMT2A 518/4885MAPT 2788/4885
US-20210102165-A1 METHODS FOR PREPARING CELLS FOR ADOPTIVE T CELL THERAPY CD4, ICOS, CD2 MEN1 3640/4885KMT2A 1396/4885MAPT 2971/4885
US-20090253691-A1 TRISUBSTITUTED 1,2,4-TRIAZOLES CHRNA1, CHRNA5, CHRNA3 MEN1 4501/4885KMT2A 1945/4885MAPT 1731/4885
US-20210163599-A1 PD-L1 BINDING AFFIMERS, AND USES RELATED THERETO PDCD1LG2, CD274, PDCD1 MEN1 3444/4885KMT2A 2041/4885MAPT 1541/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.