SCHEMBL8844679

SCHEMBL8844679

NCc1cccnc1C1CCN(Cc2ccccc2)C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.46
CYP2C9 P11712 1/20 0.46
KDM4E B2RXH2 1/20 0.45
NPC1 O15118 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
CYP2D6 P10635 2/20 0.44
USP30 Q70CQ3 2/20 0.44
ACHE P22303 3/20 0.43
CXCR4 P61073 3/20 0.43
BCHE P06276 2/20 0.43
BACE1 P56817 2/20 0.43
OPRL1 P41146 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C19 P33261 1/20 0.42
ALDH1A1 P00352 1/20 0.42
DRD2 P14416 1/20 0.41
DRD4 P21917 1/20 0.41
DRD3 P35462 1/20 0.41
CCR5 P51681 1/20 0.41
CCR3 P51677 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8844616 0.79 ACHE (0.48) CYP3A4CYP2C9KDM4ENPC1L3MBTL1
SCHEMBL1740324 0.78 CYP2D6 (0.52) CYP3A4CYP2C9CYP2D6USP30ACHE
SCHEMBL8844170 0.77 MAPK1 (0.53) L3MBTL1CYP2D6USP30ACHEBCHE
SCHEMBL19318462 0.75 DPP4 (0.41) CYP3A4CYP2D6CXCR4OPRL1
SCHEMBL8844465 0.75 PDCD1LG2 (0.52) CYP3A4CYP2C9CYP2D6USP30ACHE
SCHEMBL14868702 0.75 PDCD1LG2 (0.52) CYP3A4CYP2C9CYP2D6USP30ACHE
SCHEMBL13003294 0.75 HRH3 (0.56) KDM4EACHEBCHEBACE1DRD2
SCHEMBL9488315 0.74 MEN1 (0.49) ACHEBCHEBACE1OPRL1DRD2
Hydrochloric Acid SCHEMBL4795570 0.74 DPP4 (0.40) CYP3A4CYP2D6CXCR4OPRL1
SCHEMBL2710149 0.73 ACHE (0.57) ACHEBCHEBACE1DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5622966-A BACTERICIDES TREATING INFECTIONS WARNER-LAMBERT COMPANY (US) 1997-04-22 US disclosed
US-5446044-A Bactericides WARNER-LAMBERT COMPANY (US) 1995-08-29 US disclosed
US-5384407-A Pyrrolidine compounds WARNER-LAMBERT COMPANY (US) 1995-01-24 US disclosed
US-5342844-A 7-substituted quinolones and naphthyridones as antibacterial agents WARNER-LAMBERT COMPANY (US) 1994-08-30 US disclosed
WO-1993016077-A1 7-SUBSTITUTED QUINOLONES AND NAPHTHYRIDONES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1993-08-19 WO disclosed
US-5221676-A 7-substituted quinolones and naphthyridones as antibacterial agents WARNER-LAMBERT COMPANY (US) 1993-06-22 US disclosed