SCHEMBL8844843

SCHEMBL8844843

CC[C@](CCC(=O)O)(C(=O)OC)c1ccncc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.41
CYP19A1 P11511 3/20 0.40
CYP17A1 P05093 1/20 0.40
GAA P10253 2/20 0.40
BCHE P06276 1/20 0.39
USP2 O75604 1/20 0.36
KCNN4 O15554 1/20 0.36
ALDH1A1 P00352 4/20 0.36
ESR1 P03372 1/20 0.36
CYP3A4 P08684 1/20 0.36
ESR2 Q92731 1/20 0.36
KDM4E B2RXH2 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
PTPRB P23467 1/20 0.34
POLB P06746 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
SRC P12931 1/20 0.33
FFAR1 O14842 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8844840 1.00 TSHR (0.41) TSHRCYP19A1CYP17A1GAABCHE
SCHEMBL8844985 0.85 ALDH1A1 (0.40) TSHRCYP19A1CYP17A1GAABCHE
SCHEMBL9368728 0.76 TSHR (0.43) TSHRCYP19A1CYP17A1GAAALDH1A1
SCHEMBL16290265 0.74 CYP19A1 (0.43) TSHRCYP19A1CYP17A1ALDH1A1CYP3A4
SCHEMBL13658222 0.73 CYP19A1 (0.40) TSHRCYP19A1CYP17A1GAAALDH1A1
SCHEMBL11279155 0.71 BCHE (0.46) TSHRGAABCHEUSP2ALDH1A1
SCHEMBL27506956 0.70 ALDH1A1 (0.47) TSHRALDH1A1ESR1CYP3A4ESR2
SCHEMBL6673953 0.70 KCNN4 (0.47) GAAKCNN4CYP3A4CYP2C9CYP2C19
SCHEMBL4005855 0.70 KCNN4 (0.47) TSHRGAAKCNN4CYP3A4KDM4E
SCHEMBL28773067 0.69 ALDH1A1 (0.45) TSHRCYP19A1BCHEUSP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5661014-A Chiral compounds and their resolution synthesis using enantioselective esterases CHIROSCIENCE LIMITED (GB) 1997-08-26 US disclosed
EP-0599959-A1 CHIRAL GLUTARATE ESTERS, THEIR RESOLUTION AND DERIVED GLUTARIMIDE COMPOUNDS Chiroscience Limited (GB) 1994-06-08 EP disclosed
WO-1993004058-A1 CHIRAL GLUTARATE ESTERS, THEIR RESOLUTION AND DERIVED GLUTARIMIDE COMPOUNDS CHIROSCIENCE LIMITED (GB) 1993-03-04 WO disclosed