SCHEMBL8844985

SCHEMBL8844985

CCC(CCC(=O)O)(C(=O)O)c1ccncc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
CYP1A2 P05177 2/20 0.40
MEN1 O00255 1/20 0.40
THRB P10828 1/20 0.40
KMT2A Q03164 1/20 0.40
ESR1 P03372 1/20 0.39
CYP3A4 P08684 1/20 0.39
ESR2 Q92731 1/20 0.39
BCHE P06276 1/20 0.39
TSHR P16473 4/20 0.39
CYP19A1 P11511 2/20 0.38
CYP17A1 P05093 1/20 0.38
FFAR1 O14842 1/20 0.36
GAA P10253 2/20 0.36
MAPK1 P28482 1/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 1/20 0.35
CHEK1 O14757 1/20 0.34
FYN P06241 1/20 0.34
PDGFRB P09619 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16290265 0.86 CYP19A1 (0.43) ALDH1A1CYP1A2MEN1KMT2ACYP3A4
SCHEMBL8844843 0.85 TSHR (0.41) ALDH1A1CYP1A2ESR1CYP3A4ESR2
SCHEMBL8844840 0.85 TSHR (0.41) ALDH1A1CYP1A2ESR1CYP3A4ESR2
SCHEMBL27506956 0.85 ALDH1A1 (0.47) ALDH1A1CYP1A2MEN1THRBKMT2A
SCHEMBL11279155 0.75 BCHE (0.46) ALDH1A1CYP1A2MEN1KMT2AESR1
SCHEMBL28773067 0.73 ALDH1A1 (0.45) ALDH1A1CYP1A2MEN1THRBKMT2A
SCHEMBL11649341 0.73 ALDH1A1 (0.53) ALDH1A1CYP1A2ESR1CYP3A4ESR2
SCHEMBL9614708 0.72 ALDH1A1 (0.45) ALDH1A1MEN1KMT2AESR1CYP3A4
SCHEMBL27496397 0.72 NAPRT (0.40) ALDH1A1CYP1A2MEN1KMT2ACYP3A4
SCHEMBL28583888 0.72 ESR1 (0.46) ALDH1A1CYP1A2MEN1KMT2AESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5661014-A Chiral compounds and their resolution synthesis using enantioselective esterases CHIROSCIENCE LIMITED (GB) 1997-08-26 US disclosed
EP-0599959-A1 CHIRAL GLUTARATE ESTERS, THEIR RESOLUTION AND DERIVED GLUTARIMIDE COMPOUNDS Chiroscience Limited (GB) 1994-06-08 EP disclosed
WO-1993004058-A1 CHIRAL GLUTARATE ESTERS, THEIR RESOLUTION AND DERIVED GLUTARIMIDE COMPOUNDS CHIROSCIENCE LIMITED (GB) 1993-03-04 WO disclosed