SCHEMBL8848904

SCHEMBL8848904

COc1ccc(COCCCCCn2nnc(-c3ccc(OC(=O)C(C)(C)C)cc3)n2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.47
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
TSHR P16473 2/20 0.47
HSD17B10 Q99714 2/20 0.47
LMNA P02545 1/20 0.47
LTA4H P09960 1/20 0.47
TP53 P04637 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.44
MAPK1 P28482 1/20 0.44
USP2 O75604 1/20 0.43
MMP1 P03956 1/20 0.43
MMP2 P08253 1/20 0.43
MMP3 P08254 1/20 0.43
MMP9 P14780 1/20 0.43
MMP8 P22894 1/20 0.43
MMP13 P45452 1/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8849336 0.99 TSHR (0.47) SMN1; SMN2NPC1RAB9ATSHRHSD17B10
SCHEMBL8848700 0.92 SMN1; SMN2 (0.50) SMN1; SMN2NPC1RAB9ATSHRHSD17B10
SCHEMBL8849188 0.89 MAPK1 (0.52) SMN1; SMN2NPC1RAB9ATSHRL3MBTL1
SCHEMBL8848714 0.87 HSD17B10 (0.51) SMN1; SMN2NPC1RAB9ATSHRHSD17B10
SCHEMBL8848642 0.86 HSD17B10 (0.52) SMN1; SMN2NPC1RAB9ATSHRHSD17B10
SCHEMBL8848658 0.85 TP53 (0.45) SMN1; SMN2RAB9ATSHRHSD17B10LMNA
SCHEMBL8848912 0.84 LTA4H (0.54) SMN1; SMN2NPC1RAB9ATSHRHSD17B10
SCHEMBL8848405 0.82 NPC1 (0.64) SMN1; SMN2NPC1RAB9ATSHRHSD17B10
SCHEMBL8848828 0.82 LTA4H (0.47) SMN1; SMN2NPC1RAB9ATSHRHSD17B10
SCHEMBL8848588 0.81 LTA4H (0.48) SMN1; SMN2NPC1RAB9ATSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5602161-A ELASTASE INHIBITORS; PREVENTING AND TREATING EMPHYSEMA, ENDOTOXIN-INDUCED LUNG DISORDERS WAKAMOTO PHARMACEUTICAL CO., LTD. (JP) 1997-02-11 US disclosed
EP-0676396-A1 Tetrazolylphenyl pivalate derivatives and medicinal composition containing the same as effective component Wakamoto Pharmaceutical Co., Ltd. (JP) 1995-10-11 EP disclosed