SCHEMBL8851148

SCHEMBL8851148

COC(=O)c1ccc2cccc(C(C)C)cc1-2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 4/20 0.49
SLC6A4 P31645 3/20 0.49
SLC6A2 P23975 1/20 0.49
RXRA P19793 1/20 0.48
RXRB P28702 1/20 0.48
RXRG P48443 1/20 0.48
KDM4E B2RXH2 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
GABRA1 P14867 2/20 0.42
GABRG2 P18507 2/20 0.42
GABRB3 P28472 2/20 0.42
GABRA3 P34903 2/20 0.42
ALDH1A1 P00352 3/20 0.41
MEN1 O00255 2/20 0.41
MAPT P10636 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20173749 0.91 SLC6A3 (0.49) SLC6A3SLC6A4SLC6A2KDM4EGABRA1
SCHEMBL10415503 0.83 RXRA (0.59) RXRARXRBRXRGKDM4EHDAC4
SCHEMBL10414624 0.83 RXRA (0.51) RXRARXRBRXRGKDM4EHDAC4
SCHEMBL20173748 0.82 NR4A2 (0.51) KDM4EGABRA1GABRG2GABRB3GABRA3
SCHEMBL10414622 0.81 SLC6A3 (0.57) SLC6A3SLC6A4SLC6A2KDM4ECYP1A2
SCHEMBL6698627 0.81 CYP46A1 (0.50) SLC6A3SLC6A4SLC6A2KDM4ECYP1A2
SCHEMBL13524622 0.78 RXRA (0.51) SLC6A3SLC6A4SLC6A2RXRARXRB
SCHEMBL29978969 0.78 SLC6A3 (0.71) SLC6A3SLC6A4SLC6A2KDM4ECYP1A2
SCHEMBL6797969 0.78 SLC6A3 (0.71) SLC6A3SLC6A4SLC6A2KDM4ECYP1A2
SCHEMBL24579589 0.78 SLC6A3 (0.49) SLC6A3SLC6A4SLC6A2GABRA1GABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-9077694-A None JP disclosed
JP-H0977694-A NEW PRODUCTION OF GUAIAZULENE OR ITS DERIVATIVE TAKASAGO INTERNATL CORP 1997-03-25 JP disclosed
US-4912134-A Methyl ester substitution AJINOMOTO COMPANY, INC. (JP) 1990-03-27 US disclosed
US-4859701-A Azulene derivatives and pharmaceutical compositions containing them AJINOMOTO CO., INC. (JP) 1989-08-22 US disclosed
EP-0266956-A2 Azulene derivatives and pharmaceutical compositions containing them AJINOMOTO CO., INC. (JP) 1988-05-11 EP disclosed