SCHEMBL8854

SCHEMBL8854

COc1cc(COC=O)cc(OC)c1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.46
CYP1A1 P04798 1/20 0.41
CYP1B1 Q16678 1/20 0.41
CYP19A1 P11511 1/20 0.40
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
POLB P06746 1/20 0.39
ERN1 O75460 1/20 0.39
ABCB1 P08183 1/20 0.38
CALM1 P0DP23 2/20 0.38
AKR1B1 P15121 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC8 Q9BY41 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1828440 0.81 IDO1 (0.61) KMT2AMEN1
SCHEMBL6342 0.79 IDO1 (0.55) ALDH1A1POLBCALM1
Iodide SCHEMBL9356671 0.78 IDO1 (0.53) ALDH1A1POLBCALM1
SCHEMBL28560899 0.78 IDO1 (0.53) ALDH1A1POLBCALM1
SCHEMBL28552476 0.78 IDO1 (0.53) ALDH1A1POLBCALM1
SCHEMBL17368761 0.77 PTGS2 (0.44) ALDH1A1CYP1A1CYP1B1CYP19A1CALM1
SCHEMBL17304947 0.76 ALDH1A1 (0.42) ALDH1A1KMT2AMEN1
SCHEMBL8395 0.76 PTGS2 (0.53) CYP19A1KMT2AMEN1ABCB1
SCHEMBL2093141 0.76 ERN1 (0.49) ALDH1A1CYP1A1CYP1B1ERN1
SCHEMBL1162423 0.76 ALDH1A1 (0.52) ALDH1A1CYP1A1CYP1B1CYP19A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2555 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3053944-B1 METHOD FOR PRODUCING POLYALKYLENE GLYCOL DERIVATIVE HAVING AMINO GROUP AT END, POLYMERIZATION INITIATOR FOR USE IN THE SAME, AND ALCOHOL COMPOUND AS RAW MATERIAL FOR THE POLYMERIZATION INITIATOR SHINETSU CHEMICAL CO (JP) 2021-10-06 EP claimed
US-20210300932-A1 CYCLIC PEPTIDES TARGETING ALPHA-4-BETA-7 INTEGRIN ZEALAND PHARMA A/S (DK) 2021-09-30 US claimed
US-11072616-B2 Cyclic peptides targeting alpha-4-beta-7 integrin UNIVERSITE DE MONTREAL (CA) 2021-07-27 US claimed
WO-2020022892-A1 TUBULYSIN DERIVATIVES AND METHODS FOR PREPARING THE SAME RIJKSUNIVERSITEIT GRONINGEN (NL) 2020-01-30 WO claimed
US-8618286-B2 Benzoxazines, benzothiazines, and related compounds having NOS inhibitory activity NEURAXON, INC. (CA) 2013-12-31 US claimed
EP-2098508-B1 Processes for preparing cyclic derivatives which are modulators of chemokine receptor activity BRISTOL MYERS SQUIBB CO (US) 2012-06-20 EP claimed
US-8106043-B2 Benzoxazines, benzothiazines, and related compounds having NOS inhibitory activity NEURAXON, INC. (CA) 2012-01-31 US claimed
US-6677372-B2 N-(3-benzofuranyl)urea-derivatives BAYER AKTIENGESELLSCHAFT (DE) 2004-01-13 US claimed
EP-0882024-B1 RETROVIRAL PROTEASE INHIBITING COMPOUNDS ABBOTT LAB (US) 2002-02-06 EP claimed
US-5709848-A COMPOUNDS FOR COSMETICS FOR SKINS L'OREAL (FR) 1998-01-20 US claimed
EP-0220923-B1 Dipeptides and process GRACE W R & CO (US) 1994-04-27 EP claimed
EP-0170280-B1 NOVEL INTERMEDIATES AND PROCESS FOR THE PREPARATION OF 3-ACYLAMINO-1-HYDROXY-2-AZETIDINONES E.R. Squibb & Sons, Inc. (US) 1990-12-05 EP claimed
EP-0362634-A2 Basic dihydropyridines, process for their preparation and their use as intermediates BAYER AG (DE) 1990-04-11 EP claimed
US-4810817-A ARTIFICIAL SWEETENERS W. R. GRACE & CO. (US) 1989-03-07 US claimed
US-4710583-A ENZYMATIC COUPLING OF PHENYLSERINE WITH ASPARTIC ACID; HYDROGENATION W. R. GRACE & CO. (US) 1987-12-01 US claimed
EP-0220923-A2 Dipeptides and process W.R. Grace & Co.-Conn. (US) 1987-05-06 EP claimed
US-4581170-A N-hydroxyl protecting groups and process and intermediates for the preparation of 3-acylamino-1-hydroxy-2-azetidinones E. R. SQUIBB & SONS, INC. (US) 1986-04-08 US claimed
EP-0170280-A1 Novel intermediates and process for the preparation of 3-acylamino-1-hydroxy-2-azetidinones E.R. Squibb & Sons, Inc. (US) 1986-02-05 EP claimed
US-4119493-A IN PRESENCE OF METALLOPROTEINASE ENZYME (ZAIDANHOJIN) SAGAMI CHEMICAL RESEARCH CENTER (JP) 1978-10-10 US claimed
US-4113867-A ANTHELMINTICS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1978-09-12 US claimed