SCHEMBL8856892

SCHEMBL8856892

COc1ccc2c(c1NS(C)(=O)=O)CCCC2C#N

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
ADRA2A P08913 4/20 0.40
ADRA1A P35348 6/20 0.39
MEN1 O00255 1/20 0.39
ALOX15 P16050 1/20 0.39
KMT2A Q03164 1/20 0.39
HSD11B1 P28845 1/20 0.36
HSD17B2 P37059 1/20 0.36
TAS1R3 Q7RTX0 2/20 0.35
TAS1R1 Q7RTX1 2/20 0.35
TAS1R2 Q8TE23 2/20 0.35
CYP17A1 P05093 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9814140 0.77 PARP1 (0.49) CA1CA2ADRA1A
SCHEMBL8857004 0.76 ADRA1A (0.43) CA1CA2ADRA1A
SCHEMBL10751929 0.76 ADRA1A (0.40) CA1CA2ADRA1ATAS1R3TAS1R1
SCHEMBL9814134 0.75 CA1 (0.51) CA1CA2HSD11B1TAS1R3TAS1R1
SCHEMBL8857197 0.74 NPSR1 (0.42) CA1CA2ADRA1AMEN1KMT2A
SCHEMBL7101744 0.73 ADRA2A (0.48) CA1CA2ADRA2AADRA1AMEN1
SCHEMBL8856947 0.73 ADRA1A (0.74) ADRA2AADRA1AMEN1ALOX15KMT2A
Hydrochloric Acid SCHEMBL7104810 0.72 ADRA2A (0.48) CA1CA2ADRA2AADRA1AMEN1
SCHEMBL7098679 0.72 ADRA2A (0.48) ADRA2AADRA1AMEN1ALOX15KMT2A
SCHEMBL20478812 0.70 ADRA1A (0.49) ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5610174-A Use of α1A -selective adrenoceptor agonists for the treatment of urinary incontinence SYNAPTIC PHARMACEUTICAL CORPORATION (US) 1997-03-11 US disclosed
US-4634705-A Adrenergic amidines ABBOTT LABORATORIES (US) 1987-01-06 US disclosed