SCHEMBL8858100

SCHEMBL8858100

CCOC(=O)CC(C(=O)OCC)N1CCN(CC2CN(C3CCN(C)CC3)C(=O)O2)CC1.CN1CCC(N2CC(COS(C)(=O)=O)OC2=O)CC1

nearest known ligand 0.41

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 4/20 0.41
ITGB3 P05106 1/20 0.35
ITGA2B P08514 1/20 0.35
CYP2D6 P10635 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8858105 0.93 HTR2B (0.40) HTR2BITGB3ITGA2BCYP2D6
SCHEMBL7306776 0.93 HTR2B (0.46) HTR2BITGB3ITGA2BCYP2D6
SCHEMBL8858148 0.86 ITGB3 (0.35) HTR2BITGB3ITGA2B
SCHEMBL7311868 0.85 HTR2B (0.46) HTR2BITGB3ITGA2BCYP2D6
SCHEMBL7304230 0.82 HTR2B (0.43) HTR2BITGB3ITGA2BCYP2D6
SCHEMBL8858104 0.82 ITGB3 (0.34) HTR2BITGB3ITGA2BCYP2D6
SCHEMBL8858116 0.82 KDM4E (0.35) HTR2BITGB3ITGA2B
SCHEMBL8858110 0.82 ITGB3 (0.34) HTR2BITGB3ITGA2B
SCHEMBL8858160 0.82 ITGB3 (0.34) HTR2BITGB3ITGA2BCYP2D6
SCHEMBL8858159 0.81 ITGB3 (0.34) HTR2BITGB3ITGA2BCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5627197-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-05-06 US disclosed