SCHEMBL7306776

SCHEMBL7306776

CCOC(=O)CC(C(=O)OCC)N1CCN(CC2CN(C3CCN(C)CC3)C(=O)O2)CC1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 6/20 0.46
ITGB3 P05106 1/20 0.39
ITGA2B P08514 1/20 0.39
CYP2D6 P10635 1/20 0.35
MAPT P10636 1/20 0.31
MAPK1 P28482 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
LMNA P02545 1/20 0.31
CACNA2D1 P54289 1/20 0.31
CACNA1B Q00975 1/20 0.31
CACNB1 Q02641 1/20 0.31
CACNA1C Q13936 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8858100 0.93 HTR2B (0.41) HTR2BITGB3ITGA2BCYP2D6
SCHEMBL7311868 0.92 HTR2B (0.46) HTR2BITGB3ITGA2BCYP2D6MAPT
SCHEMBL7304230 0.89 HTR2B (0.43) HTR2BITGB3ITGA2BCYP2D6L3MBTL1
SCHEMBL8858105 0.85 HTR2B (0.40) HTR2BITGB3ITGA2BCYP2D6
SCHEMBL7313564 0.84 ITGB3 (0.39) HTR2BITGB3ITGA2BCYP2D6MAPT
SCHEMBL7313518 0.82 HTR2B (0.38) HTR2BITGB3ITGA2BLMNA
SCHEMBL7315163 0.79 ITGB3 (0.38) HTR2BITGB3ITGA2BCYP2D6MAPT
SCHEMBL7308256 0.79 ITGB3 (0.38) HTR2BITGB3ITGA2BCYP2D6MAPT
SCHEMBL7313170 0.79 ITGB3 (0.38) HTR2BITGB3ITGA2BCYP2D6MAPT
SCHEMBL7309903 0.78 ITGB3 (0.38) HTR2BITGB3ITGA2BCYP2D6MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0727425-A1 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1996-08-21 EP disclosed