SCHEMBL8858771

SCHEMBL8858771

CC(C)(C)OC(=O)N1CCc2nc(-c3ccc(C(=O)O)cc3)sc2CC1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
GRAMD1A Q96CP6 1/20 0.46
GPR119 Q8TDV5 9/20 0.44
HDAC4 P56524 1/20 0.41
ADORA1 P30542 1/20 0.41
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
FGFR3 P22607 1/20 0.40
KDR P35968 1/20 0.40
TBK1 Q9UHD2 1/20 0.40
PTGER4 P35408 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8858696 0.93 GRAMD1A (0.55) NPC1RAB9AGRAMD1AADORA1KDM4E
SCHEMBL8858814 0.88 NPC1 (0.47) NPC1RAB9AGRAMD1AGPR119ADORA1
SCHEMBL8858740 0.82 HDAC4 (0.49) NPC1RAB9AGRAMD1AGPR119HDAC4
SCHEMBL3586943 0.82 NPC1 (0.43) NPC1RAB9AGRAMD1AGPR119FGFR3
SCHEMBL3666966 0.81 NPC1 (0.54) NPC1RAB9AGRAMD1AADORA1KDM4E
SCHEMBL15166579 0.81 ESR2 (0.50) NPC1RAB9AGRAMD1AADORA1KDM4E
SCHEMBL8858785 0.81 HDAC4 (0.49) NPC1RAB9AGRAMD1AGPR119HDAC4
SCHEMBL20792856 0.80 DPP4 (0.53) NPC1RAB9AGRAMD1AADORA1KDM4E
SCHEMBL10097946 0.80 MKNK1 (0.48) NPC1RAB9AGRAMD1AADORA1KDM4E
SCHEMBL8858610 0.80 NPC1 (0.53) NPC1RAB9AGRAMD1AADORA1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607944-A ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-03-04 US disclosed
EP-0639575-A1 Bicyclic heterocycles, medicaments comprising these compounds and processes for their production Dr. Karl Thomae GmbH (DE) 1995-02-22 EP disclosed