SCHEMBL8858740

SCHEMBL8858740

CC(C)(C)OC(=O)N1CCc2nc(-c3ccc(C(=O)N[C@H]4CC[C@H](C(=O)O)CC4)cc3)sc2CC1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 3/20 0.49
HDAC6 Q9UBN7 2/20 0.44
GRAMD1A Q96CP6 1/20 0.44
POLB P06746 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41
GPR119 Q8TDV5 6/20 0.41
USP30 Q70CQ3 3/20 0.41
PTPN2 P17706 1/20 0.39
PTPN1 P18031 1/20 0.39
PTPN6 P29350 1/20 0.39
KDM4E B2RXH2 1/20 0.39
PKM P14618 1/20 0.39
DRD3 P35462 1/20 0.39
RIPK2 O43353 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8858733 0.94 GRAMD1A (0.51) HDAC4HDAC6GRAMD1ANPC1RAB9A
SCHEMBL8858785 0.93 HDAC4 (0.49) HDAC4HDAC6GRAMD1APOLBNPC1
SCHEMBL8858682 0.87 GRAMD1A (0.51) HDAC4HDAC6GRAMD1ANPC1RAB9A
SCHEMBL8858794 0.86 HDAC4 (0.43) HDAC4HDAC6NPC1RAB9AKMT2A
SCHEMBL8858634 0.84 USP30 (0.49) HDAC4GRAMD1APOLBNPC1RAB9A
SCHEMBL8858824 0.83 GRAMD1A (0.47) HDAC4GRAMD1ANPC1RAB9AGPR119
SCHEMBL8858771 0.82 NPC1 (0.47) HDAC4GRAMD1ANPC1RAB9AGPR119
SCHEMBL8858804 0.79 HDAC4 (0.42) HDAC4HDAC6NPC1RAB9AKMT2A
SCHEMBL8858775 0.78 MEN1 (0.43) HDAC4HDAC6NPC1RAB9AKMT2A
SCHEMBL8858741 0.78 SCN4A (0.41) GRAMD1APOLBPTPN2PTPN1PTPN6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607944-A ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-03-04 US disclosed
EP-0639575-A1 Bicyclic heterocycles, medicaments comprising these compounds and processes for their production Dr. Karl Thomae GmbH (DE) 1995-02-22 EP disclosed