SCHEMBL8860266

SCHEMBL8860266

O=C1c2ccccc2C(=O)N1[CH]Cc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 2/20 0.46
TDP1 Q9NUW8 2/20 0.44
L3MBTL1 Q9Y468 3/20 0.43
MAOB P27338 2/20 0.43
ALDH1A1 P00352 3/20 0.42
NR1H3 Q13133 2/20 0.42
NR1H2 P55055 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
GAA P10253 1/20 0.42
CA12 O43570 1/20 0.41
CA9 Q16790 1/20 0.41
ALDH2 P05091 1/20 0.41
CHRM1 P11229 1/20 0.41
CES1 P23141 1/20 0.41
ALDH3A1 P30838 1/20 0.41
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10421305 0.81 MAOB (0.50) CASP3TDP1L3MBTL1MAOBALDH1A1
SCHEMBL10421307 0.81 MAOB (0.50) CASP3TDP1L3MBTL1MAOBALDH1A1
SCHEMBL23830079 0.81 MAOB (0.50) CASP3TDP1L3MBTL1MAOBALDH1A1
SCHEMBL27338871 0.75 CA12 (0.44) CASP3ALDH1A1NR1H3GAACA12
SCHEMBL6329301 0.75 DRD3 (0.43) CASP3TDP1ALDH1A1MEN1KMT2A
SCHEMBL5190685 0.75 ALDH1A1 (0.44) CASP3ALDH1A1GAACA12CA9
SCHEMBL2183011 0.75 CASP3 (0.40) CASP3ALDH1A1MEN1KMT2AGAA
SCHEMBL28119261 0.73 CASP3 (0.55) CASP3ALDH1A1MEN1KMT2ACA12
SCHEMBL5177139 0.72 DRD3 (0.44) CASP3ALDH1A1NR1H3NR1H2MEN1
SCHEMBL8498912 0.72 CASP3 (0.44) CASP3TDP1L3MBTL1MAOBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5698698-A Process for preparation of N-tert.butyl-decahydro-2- 2(R)-hydroxy-4-phenyl-3(S)-phthalimidobutyl!-(4aS,8aS)-isoquinoline-3(S)-carboxamide HOFFMANN-LA ROCHE INC. (US) 1997-12-16 US disclosed
US-5502210-A 1H-isoindole-1,3-dione compounds HOFFMANN-LA ROCHE INC. (US) 1996-03-26 US disclosed