SCHEMBL8861902

SCHEMBL8861902

Cc1ccc(CN2CCN(Cc3n[nH]cc3-c3ccccc3C)C(C)C2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH2 P25021 1/20 0.42
POLB P06746 2/20 0.40
LMNA P02545 1/20 0.40
MAPK1 P28482 2/20 0.39
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39
BACE1 P56817 1/20 0.39
ALDH1A1 P00352 2/20 0.38
MET P08581 1/20 0.37
AXL P30530 1/20 0.37
MERTK Q12866 1/20 0.37
MAPT P10636 2/20 0.37
TP53 P04637 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
GAA P10253 2/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8861849 0.94 HRH2 (0.46) HRH2POLBLMNACYP2D6CYP2C19
SCHEMBL9047699 0.79 LMNA (0.48) POLBLMNAALDH1A1MAPTDRD2
SCHEMBL14528083 0.69 HRH2 (0.66) HRH2POLBLMNAACHEMAPT
SCHEMBL5692251 0.69 HRH2 (0.66) HRH2POLBLMNAACHEMAPT
SCHEMBL20284487 0.69 HRH2 (0.66) HRH2POLBLMNAACHEMAPT
SCHEMBL9039441 0.68 LMNA (0.52) POLBLMNAMAPK1ALDH1A1DRD2
SCHEMBL8861842 0.64 SIGMAR1 (0.53) POLBLMNAALDH1A1MAPTCYP2D6
SCHEMBL20432883 0.64 LMNA (0.71) POLBLMNAMAPK1BCHEACHE
SCHEMBL20432817 0.63 KDM4E (0.43) HRH2POLBLMNAMAPK1ALDH1A1
SCHEMBL13554190 0.62 HRH2 (0.56) HRH2ACHEALDH1A1MAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5684006-A Isoxazole and pyrazole derivatives as dopamine receptor subtype ligands MERCK, SHARP & DOHME, LTD. (GB) 1997-11-04 US disclosed