SCHEMBL8864090

SCHEMBL8864090

NC(=O)OCC1CCc2ccccc2O1

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.63
HTR1A P08908 5/20 0.44
SIGMAR1 Q99720 2/20 0.44
ADRA2A P08913 1/20 0.44
ADRA2B P18089 1/20 0.44
ADRA2C P18825 1/20 0.44
SLC6A4 P31645 1/20 0.43
PTGDR Q13258 1/20 0.43
HTR1D P28221 3/20 0.42
L3MBTL1 Q9Y468 2/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27285788 0.81 CA2 (0.54) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL406490 0.81 CA2 (0.56) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL1520875 0.80 CA2 (0.67) CA2HTR1ASIGMAR1ADRA2AADRA2B
Bicarbonate SCHEMBL6086499 0.78 CA2 (0.56) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL30711451 0.77 CA2 (0.62) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL5274616 0.77 CA2 (1.00) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL3975518 0.77 CA2 (0.62) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL9536357 0.76 ALOX5 (0.63) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL16428909 0.76 CA2 (0.54) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL15211143 0.76 CA2 (0.54) CA2HTR1ASIGMAR1ADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1038032-C {(Benzodioxan, benzofuran or benzopyran) alkylamino} alkyl substituted guanidines JANSSEN PHARMACEUTICA NV (BE) 1998-04-15 CN disclosed
US-5703115-A VASOCONSTRICTORS JANSSEN PHARMACEUTICA, N.V. (BE) 1997-12-30 US disclosed
US-5688952-A VASOCONSTRICTOR INTERMEDIATES JANSSEN PHARMACEUTICA, N.V. (BE) 1997-11-18 US disclosed
CN-1079470-A [(benzo two  alkane, cumarone or chromene) alkylamino] alkyl substituted guanidines JANSSEN PHARMACEUTICA NV (BE) 1993-12-15 CN disclosed