SCHEMBL8864634

SCHEMBL8864634

CC1=NC(c2cc(C)cs2)c2ccccc2CN1C

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.40
SLC6A2 P23975 16/20 0.36
SLC6A4 P31645 16/20 0.36
SLC6A3 Q01959 15/20 0.36
PTGS2 P35354 1/20 0.35
CYP2D6 P10635 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8865110 0.71 SLC6A2 (0.52) KCNH2SLC6A2SLC6A4SLC6A3
SCHEMBL8864666 0.71 KCNH2 (0.55) KCNH2SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL8864617 0.69 KCNH2 (0.52) KCNH2SLC6A2SLC6A4SLC6A3
SCHEMBL9257287 0.63 MEN1 (0.37) SMN1; SMN2
Hydrochloric Acid SCHEMBL8556675 0.60 MAOA (0.42) KCNH2CYP2D6SMN1; SMN2
SCHEMBL12539165 0.60 PLG (0.41) PTGS2
SCHEMBL8558645 0.59 KCNH2 (0.72) KCNH2SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL8555627 0.59 KCNH2 (0.72) KCNH2SLC6A2SLC6A4SLC6A3CYP2D6
Hydrochloric Acid SCHEMBL8557094 0.59 KCNH2 (0.60) KCNH2SLC6A2SLC6A4SLC6A3PTGS2
SCHEMBL8557530 0.59 KCNH2 (0.72) KCNH2SLC6A2SLC6A4SLC6A3CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5624922-A Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1997-04-29 US disclosed
EP-0597540-B1 Aryl-fused and hetaryl-fused-2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC (US) 1996-06-05 EP disclosed
US-5380721-A Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1995-01-10 US disclosed
EP-0597540-A1 Aryl-fused and hetaryl-fused-2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1994-05-18 EP disclosed