SCHEMBL8865110

SCHEMBL8865110

CC1=NC(c2ccc(Cl)cc2)c2ccccc2CN1C

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 7/20 0.52
SLC6A4 P31645 7/20 0.52
SLC6A3 Q01959 7/20 0.52
KCNH2 Q12809 3/20 0.51
NOS3 P29474 1/20 0.40
PRCP P42785 1/20 0.39
HTR2A P28223 4/20 0.38
HTR2C P28335 4/20 0.38
HTR2B P41595 4/20 0.38
HRH3 Q9Y5N1 4/20 0.38
GAA P10253 2/20 0.38
KMT2A Q03164 1/20 0.38
SCN5A Q14524 1/20 0.37
KDM4E B2RXH2 1/20 0.37
NPC1 O15118 1/20 0.37
ALDH1A1 P00352 1/20 0.37
RAB9A P51151 1/20 0.37
MAOB P27338 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8864617 0.83 KCNH2 (0.52) SLC6A2SLC6A4SLC6A3KCNH2GAA
SCHEMBL8557736 0.79 KCNH2 (0.83) SLC6A2SLC6A4SLC6A3KCNH2NOS3
SCHEMBL8554225 0.77 KCNH2 (0.83) SLC6A2SLC6A4SLC6A3KCNH2HTR2A
Hydrochloric Acid SCHEMBL8864724 0.76 KCNH2 (0.54) SLC6A2SLC6A4SLC6A3KCNH2NOS3
SCHEMBL11018524 0.71 HTR2A (0.44) SLC6A2SLC6A4SLC6A3KCNH2NOS3
SCHEMBL8864634 0.71 KCNH2 (0.40) SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL8864666 0.71 KCNH2 (0.55) SLC6A2SLC6A4SLC6A3KCNH2KDM4E
Hydrochloric Acid SCHEMBL8557094 0.71 KCNH2 (0.60) SLC6A2SLC6A4SLC6A3KCNH2NOS3
SCHEMBL8558645 0.71 KCNH2 (0.72) SLC6A2SLC6A4SLC6A3KCNH2PRCP
SCHEMBL8555627 0.71 KCNH2 (0.72) SLC6A2SLC6A4SLC6A3KCNH2PRCP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5624922-A Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1997-04-29 US disclosed
EP-0597540-B1 Aryl-fused and hetaryl-fused-2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC (US) 1996-06-05 EP disclosed
US-5380721-A Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1995-01-10 US disclosed
EP-0597540-A1 Aryl-fused and hetaryl-fused-2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1994-05-18 EP disclosed