SCHEMBL8864698

SCHEMBL8864698

CN1Cc2ccccc2C(c2ccccc2)N=C1CCc1ccc(N)cc1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 8/20 0.83
MAOB P27338 4/20 0.41
MAOA P21397 2/20 0.41
SLC6A2 P23975 2/20 0.38
SLC6A4 P31645 2/20 0.38
SLC6A3 Q01959 2/20 0.38
SCN5A Q14524 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
NPC1 O15118 1/20 0.37
GAA P10253 1/20 0.37
RAB9A P51151 1/20 0.37
HTR6 P50406 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
CHRM2 P08172 1/20 0.34
CHRM1 P11229 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34
CHRM3 P20309 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8864716 0.99 KCNH2 (0.81) KCNH2MAOBMAOASLC6A2SLC6A4
SCHEMBL8556398 0.91 KCNH2 (1.00) KCNH2SLC6A2SLC6A4SLC6A3SCN5A
SCHEMBL8554712 0.91 KCNH2 (1.00) KCNH2SLC6A2SLC6A4SLC6A3SCN5A
SCHEMBL8555810 0.91 KCNH2 (1.00) KCNH2SLC6A2SLC6A4SLC6A3SCN5A
Hydrochloric Acid SCHEMBL8865195 0.88 KCNH2 (0.65) KCNH2SLC6A2SLC6A4SLC6A3SCN5A
Hydrochloric Acid SCHEMBL8864606 0.88 KCNH2 (0.64) KCNH2MAOBMAOASLC6A2SLC6A4
SCHEMBL8553316 0.88 KCNH2 (0.83) KCNH2MAOBSLC6A2SLC6A4SLC6A3
SCHEMBL8554225 0.88 KCNH2 (0.83) KCNH2SLC6A2SLC6A4SLC6A3SCN5A
SCHEMBL8554877 0.84 KCNH2 (0.77) KCNH2SCN5A
SCHEMBL9255302 0.84 KCNH2 (0.81) KCNH2SIGMAR1HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5624922-A Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1997-04-29 US disclosed
EP-0597540-B1 Aryl-fused and hetaryl-fused-2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC (US) 1996-06-05 EP disclosed
US-5380721-A Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1995-01-10 US disclosed
EP-0597540-A1 Aryl-fused and hetaryl-fused-2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1994-05-18 EP disclosed