SCHEMBL8865798

SCHEMBL8865798

COC(=O)Cc1cn(Cc2ccccc2)cn1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 1/20 0.54
CDK5R1 Q15078 1/20 0.54
ADRB1 P08588 1/20 0.47
ADRB3 P13945 1/20 0.47
KDM5A P29375 1/20 0.46
KDM4C Q9H3R0 1/20 0.46
KDM5B Q9UGL1 1/20 0.46
CYP11B1 P15538 1/20 0.45
CYP11B2 P19099 1/20 0.45
HPGDS O60760 1/20 0.44
CYP2E1 P05181 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2A6 P11509 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2B6 P20813 1/20 0.43
CYP2C19 P33261 1/20 0.43
TRHDE Q9UKU6 1/20 0.43
RBP4 P02753 1/20 0.41
KLKB1 P03952 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8865591 0.88 CDK5 (0.42) CDK5CDK5R1ADRB1ADRB3KDM5A
SCHEMBL8455536 0.86 ALDH1A1 (0.49) CDK5CDK5R1ADRB1ADRB3KDM5A
SCHEMBL7399708 0.84 KDM4C (0.51) CDK5CDK5R1ADRB1ADRB3KDM5A
Hydrochloric Acid SCHEMBL8762068 0.82 KDM4C (0.50) CDK5CDK5R1ADRB1ADRB3KDM5A
SCHEMBL10283948 0.82 HMOX1 (0.44) CDK5CDK5R1ADRB1ADRB3CYP11B1
SCHEMBL8344061 0.82 ALDH1A1 (0.50) CDK5CDK5R1CYP3A4CYP2D6CYP2C9
SCHEMBL6527840 0.78 CDK5 (0.47) CDK5CDK5R1ADRB1ADRB3KDM5A
SCHEMBL6069460 0.78 CDK5 (0.47) CDK5CDK5R1ADRB1ADRB3KDM5A
SCHEMBL18367381 0.77 CDK5 (0.53) CDK5CDK5R1KDM5AKDM4CKDM5B
Hydrochloric Acid SCHEMBL7356305 0.77 CDK5 (0.46) CDK5CDK5R1ADRB1ADRB3KDM5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5652257-A ANTICARCINOGENIC MERCK & CO., INC. (US) 1997-07-29 US disclosed
WO-1996010034-A2 THIOL-FREE INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1996-04-04 WO disclosed