SCHEMBL8866149

SCHEMBL8866149

NC(Cc1ccc(O)cc1)(OC(=O)/C=C/C(=O)OC(N)(Cc1ccc(O)cc1)c1ccc(O)cc1)c1ccc(O)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BLM P54132 1/20 0.45
ESR1 P03372 6/20 0.42
ESR2 Q92731 5/20 0.42
CA12 O43570 3/20 0.37
CA7 P43166 3/20 0.37
CA9 Q16790 3/20 0.37
CA14 Q9ULX7 3/20 0.37
CA4 P22748 2/20 0.37
CA6 P23280 2/20 0.37
CA5A P35218 2/20 0.37
CA5B Q9Y2D0 2/20 0.37
CA1 P00915 2/20 0.37
MET P08581 1/20 0.37
CA2 P00918 3/20 0.37
IDO1 P14902 2/20 0.35
KIF11 P52732 1/20 0.35
CAMK2A Q9UQM7 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
AKR1B10 O60218 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8866615 0.93 BLM (0.45) BLMESR1ESR2CA12CA7
Acetic Acid SCHEMBL8866221 0.66 BLM (0.62) BLMESR1ESR2CA2CAMK2A
SCHEMBL7387615 0.65 BLM (0.67) BLMESR1ESR2CA2IDO1
SCHEMBL5329248 0.65 ESR1 (0.64) BLMESR1ESR2MEN1KMT2A
SCHEMBL23963227 0.65 BLM (0.47) BLMESR1ESR2CA2IDO1
SCHEMBL20342303 0.65 BLM (0.47) BLMESR1ESR2CA2IDO1
SCHEMBL21142143 0.65 KIF11 (0.45) BLMESR1ESR2CA12CA7
SCHEMBL27747412 0.65 BLM (0.56) BLMESR1ESR2CA2IDO1
SCHEMBL28966331 0.64 BLM (0.65) BLMESR1ESR2CA2IDO1
SCHEMBL17768418 0.64 BLM (0.65) BLMESR1ESR2CA2IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5605916-A Arylalkyl-amines having anticonvulsant and neuroprotective properties ASTRA AB (SE) 1997-02-25 US disclosed
US-5539120-A Arylalkyl-amines having anticonvulsant and neuroprotective properties AGENCE SPATIALE EUROPEENNE (FR) 1996-07-23 US disclosed
EP-0356035-B1 Arylkalkyl-amines and -amides having anticonvulsant and neuroprotective properties ASTRA AB (SE) 1996-03-13 EP disclosed
US-5430044-A Arylalkyl-amines and -amides having anticonvulsant and neuroprotective properties FISONS CORPORATION (GB) 1995-07-04 US disclosed
EP-0648745-A1 Arylalkylamine having anticonvulsant and neuroprotective properties Astra Aktiebolag (SE) 1995-04-19 EP disclosed
EP-0648489-A1 Arylalkylamides having neuroprotective properties FISONS CORPORATION (US) 1995-04-19 EP disclosed
US-5331007-A Arylalkyl-amines and -amides having anticonvulsant and neuroprotective properties FISONS CORPORATION (US) 1994-07-19 US disclosed
WO-1991011995-A1 ARYLALKYL-AMINES AND -AMIDES HAVING ANTICONVULSANT AND NEUROPROTECTIVE PROPERTIES FISONS CORPORATION (US) 1991-08-22 WO disclosed
EP-0356035-A2 Arylkalkyl-amines and -amides having anticonvulsant and neuroprotective properties Astra Aktiebolag (SE) 1990-02-28 EP disclosed