SCHEMBL8866839

SCHEMBL8866839

O=C(Nc1ccccc1)c1ccncc1CCO

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.51
ADRB2 P07550 1/20 0.51
HTT P42858 2/20 0.50
BCAT2 O15382 1/20 0.50
KDR P35968 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C19 P33261 1/20 0.47
NAMPT P43490 2/20 0.47
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 1/20 0.47
HPGD P15428 1/20 0.47
KMT2A Q03164 1/20 0.47
TYK2 P29597 3/20 0.46
JAK2 O60674 2/20 0.46
CYP11B2 P19099 1/20 0.46
FLT1 P17948 1/20 0.46
ROCK2 O75116 1/20 0.46
ROCK1 Q13464 1/20 0.46
NPC1 O15118 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19358958 0.88 HTT (0.53) ALDH1A1ADRB2HTTBCAT2CYP3A4
SCHEMBL1072315 0.82 ALDH1A1 (0.73) ALDH1A1ADRB2HTTBCAT2KDR
SCHEMBL6068362 0.81 ALDH1A1 (0.60) ALDH1A1HTTKDM4EHPGDKMT2A
SCHEMBL2892111 0.79 HTT (0.56) ALDH1A1HTTNAMPTKDM4EMEN1
SCHEMBL13948995 0.78 ALDH1A1 (0.70) ALDH1A1HTTCYP3A4NAMPTKDM4E
SCHEMBL16267498 0.78 KDR (0.54) ALDH1A1ADRB2KDRCYP1A2CYP2C19
SCHEMBL2899135 0.77 MEN1 (0.67) ALDH1A1HTTNAMPTKDM4EMEN1
SCHEMBL13322124 0.76 TYK2 (0.67) ALDH1A1HTTNAMPTKDM4EMEN1
SCHEMBL28072916 0.76 HTT (0.67) ALDH1A1HTTNAMPTKDM4EMEN1
SCHEMBL28072777 0.76 JAK2 (0.67) ALDH1A1HTTCYP3A4NAMPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5700941-A Octahydronaphthyridine derivatives MERCK, SHARP & DOHME, LTD. (GB) 1997-12-23 US disclosed