SCHEMBL8867016

SCHEMBL8867016

N=C(N)c1ccc2nc(-c3ccc(C(=O)O)cc3)cn2c1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.61
KDM4E B2RXH2 7/20 0.61
MEN1 O00255 2/20 0.61
KMT2A Q03164 2/20 0.61
HSP90AA1 P07900 1/20 0.61
RXFP1 Q9HBX9 1/20 0.61
NPC1 O15118 8/20 0.54
RAB9A P51151 8/20 0.54
SMN1; SMN2 Q16637 4/20 0.54
POLB P06746 3/20 0.54
GAA P10253 2/20 0.54
ALDH1A3 P47895 3/20 0.50
GLA P06280 1/20 0.48
ALDH1A2 O94788 1/20 0.48
NR4A2 P43354 1/20 0.47
MITF O75030 1/20 0.45
KDM5A P29375 1/20 0.45
KDM5C P41229 1/20 0.45
PAX8 Q06710 1/20 0.45
CLK1 P49759 4/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetic Acid SCHEMBL4952379 0.89 ALDH1A1 (0.55) ALDH1A1KDM4EMEN1KMT2AHSP90AA1
SCHEMBL4951218 0.88 ALDH1A1 (0.53) ALDH1A1KDM4EMEN1KMT2AHSP90AA1
SCHEMBL2128582 0.84 ALDH1A3 (0.57) ALDH1A1KDM4EMEN1KMT2AHSP90AA1
Trifluoroacetic Acid SCHEMBL2128057 0.84 ALDH1A3 (0.51) ALDH1A1KDM4EMEN1KMT2AHSP90AA1
Acetic Acid SCHEMBL4952485 0.84 ALDH1A3 (0.60) ALDH1A1KDM4EMEN1KMT2AHSP90AA1
SCHEMBL8866329 0.83 SUV39H2 (0.47) ALDH1A1KDM4EMEN1KMT2AHSP90AA1
SCHEMBL2129032 0.81 ALDH1A1 (0.73) ALDH1A1KDM4EMEN1KMT2AHSP90AA1
SCHEMBL8866583 0.81 ALDH1A1 (0.62) ALDH1A1KDM4EMEN1KMT2AHSP90AA1
SCHEMBL9235389 0.81 ALDH1A1 (0.53) ALDH1A1KDM4EMEN1KMT2AHSP90AA1
SCHEMBL4726717 0.81 ALDH1A1 (0.68) ALDH1A1KDM4EMEN1KMT2AHSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5614531-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-03-25 US disclosed
EP-0668278-A1 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1995-08-23 EP disclosed