SCHEMBL8868010

SCHEMBL8868010

CC(Cl)C(=O)C(=O)OC(C)(C)C

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA12 O43570 1/20 0.31
CA14 Q9ULX7 1/20 0.31
CTSK P43235 1/20 0.30
LMNA P02545 1/20 0.30
KMT2A Q03164 1/20 0.30
CYP2D6 P10635 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1089194 0.80 DGAT1 (0.36) DGAT1CA1CA2CA7CA12
SCHEMBL11374066 0.79 CA1 (0.32) DGAT1CA1CA2CA7
SCHEMBL1088727 0.77 CA1 (0.35) DGAT1CA1CA2CA7CA12
SCHEMBL7576779 0.77 LMNA (0.35) DGAT1LMNAKMT2A
SCHEMBL11387554 0.76 DGAT1 (0.33) DGAT1CA1CA2CA7CA12
SCHEMBL29488702 0.76 DGAT1 (0.33) DGAT1CA1CA2CA7CA12
SCHEMBL17094539 0.75 LMNA (0.39) DGAT1CA1CA2CA7CA12
SCHEMBL17094267 0.75 LMNA (0.39) DGAT1CA1CA2CA7CA12
SCHEMBL3183015 0.75 LMNA (0.39) DGAT1CA1CA2CA7CA12
SCHEMBL10608008 0.73 SLC7A5 (0.41) DGAT1CA1CA2CA7CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5665746-A BACTERICIDE HOFFMANN-LA ROCHE INC. (US) 1997-09-09 US disclosed
US-5594135-A BACTERICIDES HOFFMANN-LA ROCHE INC. (US) 1997-01-14 US disclosed
US-5589473-A BACTERICIDES HOFFMANN-LA ROCHE INC. (US) 1996-12-31 US disclosed
EP-0675122-A2 Mono or bicyclic DNA gyrase inhibitors F. HOFFMANN-LA ROCHE AG (CH) 1995-10-04 EP disclosed