SCHEMBL8868342

SCHEMBL8868342

COc1ccc2c(O)c(C(c3cc[c]cc3)C3CC3)c(=O)oc2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 5/20 0.49
KDM4E B2RXH2 6/20 0.43
ALDH1A1 P00352 6/20 0.43
MAPT P10636 5/20 0.43
POLB P06746 2/20 0.43
NPC1 O15118 1/20 0.43
STAT1 P42224 1/20 0.43
RAB9A P51151 1/20 0.43
LMNA P02545 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
HPGD P15428 3/20 0.41
HSD17B10 Q99714 3/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
TP53 P04637 1/20 0.41
CYP3A4 P08684 1/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
GAA P10253 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7349247 0.79 NQO1 (0.47) NQO1KDM4EALDH1A1MAPTPOLB
SCHEMBL7354182 0.76 NQO1 (0.42) NQO1KDM4EALDH1A1MAPTPOLB
SCHEMBL7354536 0.71 CYP2C9 (0.69) NQO1KDM4EALDH1A1MAPTLMNA
SCHEMBL8494601 0.71 NQO1 (0.61) NQO1KDM4EALDH1A1MAPTPOLB
SCHEMBL7350870 0.71 VKORC1 (0.67) NQO1KDM4EALDH1A1HSD17B10MEN1
SCHEMBL6276172 0.71 NQO1 (0.73) NQO1KDM4EALDH1A1MAPTPOLB
SCHEMBL7400115 0.71 ACHE (0.40) NQO1
SCHEMBL17133407 0.70 CYP2C9 (0.72) NQO1KDM4EALDH1A1MAPTLMNA
SCHEMBL8087605 0.69 NQO1 (0.69) NQO1KDM4EALDH1A1MAPTPOLB
SCHEMBL38652222 0.69 NQO1 (0.69) NQO1KDM4EALDH1A1MAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5686486-A 4-hydroxy-benzopyran-2-ones and 4-hydroxy-cycloalkyl b!pyran-2-ones useful to treat retroviral infections PHARMACIA & UPJOHN COMPANY (US) 1997-11-11 US claimed
US-5686486-A 4-hydroxy-benzopyran-2-ones and 4-hydroxy-cycloalkyl b!pyran-2-ones useful to treat retroviral infections PHARMACIA & UPJOHN COMPANY (US) 1997-11-11 US disclosed