SCHEMBL7400115

SCHEMBL7400115

COCCOCCOCCOc1ccc2c(O)c(C(c3cccc(N)c3)C3CC3)c(=O)oc2c1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.40
MAP1LC3B Q9GZQ8 1/20 0.37
MAP1LC3A Q9H492 1/20 0.37
CYP2C9 P11712 4/20 0.37
VKORC1 Q9BQB6 1/20 0.37
HDAC1 Q13547 1/20 0.36
NQO1 P15559 3/20 0.36
PRKDC P78527 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7405458 0.84 SIGMAR1 (0.36) ACHEPRKDC
SCHEMBL7405459 0.83 HDAC1 (0.34) ACHEMAP1LC3BMAP1LC3AHDAC1NQO1
SCHEMBL7400973 0.82 MAOB (0.40) ACHEMAP1LC3BMAP1LC3ANQO1
SCHEMBL7403592 0.81 NQO1 (0.36) ACHEMAP1LC3BMAP1LC3ANQO1
SCHEMBL7400677 0.79 ROCK2 (0.35) ACHE
SCHEMBL7405503 0.79 FABP1 (0.44) MAP1LC3BMAP1LC3A
SCHEMBL7359563 0.79 CYP2C9 (0.58) ACHECYP2C9VKORC1NQO1
SCHEMBL7406127 0.77 MAPT (0.31)
SCHEMBL7406916 0.75 MGAM (0.31)
SCHEMBL7354182 0.72 NQO1 (0.42) NQO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6169181-B1 HUMAN IMMUNODEFICIENCY VIRUS PROTEINASE INHIBITORS PHARMACIA & UPJOHN COMPANY 2001-01-02 US disclosed
US-5852195-A Pyranone compounds useful to treat retroviral infections PHARMACIA & UPJOHN COMPANY (US) 1998-12-22 US disclosed
EP-0758327-A1 PYRANONE COMPOUNDS USEFUL TO TREAT RETROVIRAL INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1997-02-19 EP disclosed
WO-1995030670-A2 PYRANONE COMPOUNDS USEFUL TO TREAT RETROVIRAL INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1995-11-16 WO disclosed