SCHEMBL8868359

SCHEMBL8868359

COC(=O)CNC(=O)c1ccc(C(=O)NS(=O)(=O)c2ccc(CCNC(=O)CCc3ccccc3)cc2)cn1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
P4HTM Q9NXG6 4/20 0.48
ALDH1A1 P00352 5/20 0.45
POLB P06746 3/20 0.44
RAB9A P51151 2/20 0.43
LMNA P02545 2/20 0.43
NPC1 O15118 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HIF1A Q16665 1/20 0.43
PPARA Q07869 1/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
KDM4E B2RXH2 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
PAX8 Q06710 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8868789 0.93 P4HTM (0.48) P4HTMALDH1A1POLBRAB9ALMNA
SCHEMBL8869839 0.93 P4HTM (0.46) P4HTMALDH1A1POLBRAB9ALMNA
SCHEMBL8868297 0.92 P4HTM (0.47) P4HTMALDH1A1POLBRAB9ALMNA
SCHEMBL8868937 0.91 P4HTM (0.52) P4HTMALDH1A1POLBRAB9ANPC1
SCHEMBL8869563 0.91 P4HTM (0.45) P4HTMALDH1A1POLBRAB9ALMNA
SCHEMBL8869090 0.90 ALDH1A1 (0.51) P4HTMALDH1A1POLBRAB9ALMNA
SCHEMBL8868562 0.90 P4HTM (0.51) P4HTMRAB9ANPC1SMN1; SMN2HIF1A
SCHEMBL8868236 0.90 P4HTM (0.51) P4HTMALDH1A1POLBRAB9ALMNA
SCHEMBL8868015 0.90 POLB (0.52) P4HTMALDH1A1POLBLMNASMN1; SMN2
SCHEMBL9138512 0.89 P4HTM (0.52) P4HTMALDH1A1POLBRAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607954-A Sulfonamido- and sulfonamidocarbonylpyridine-2-carboxamides and their pyridine-n-oxides, process for their preparation and their use as pharmaceuticals HOECHST AKTIENGESELLSCHAFT (DE) 1997-03-04 US disclosed