SCHEMBL8868533

SCHEMBL8868533

O=C(CCCCCBr)OCCc1ccsc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAAA Q02083 1/20 0.41
LTA4H P09960 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.40
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
TSHR P16473 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
DGKA P23743 1/20 0.40
APP P05067 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39
OPRK1 P41145 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
PTGES O14684 1/20 0.37
ALOX5 P09917 1/20 0.37
CHRM5 P08912 1/20 0.37
CHRM1 P11229 1/20 0.37
NPC1 O15118 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3091073 0.94 NAAA (0.45) NAAALTA4HL3MBTL1ALDH1A1POLB
SCHEMBL31481673 0.87 DGKA (0.58) LTA4HTSHRDGKAPTGESALOX5
SCHEMBL20538669 0.87 DGKA (0.58) LTA4HTSHRDGKAPTGESALOX5
SCHEMBL1182457 0.87 DGKA (0.58) LTA4HTSHRDGKAPTGESALOX5
SCHEMBL17578807 0.83 TDP1 (0.54) NAAAAPPTDP1ALOX5CHRM5
SCHEMBL34470938 0.80 TDP1 (0.51) NAAALTA4HL3MBTL1ALDH1A1POLB
SCHEMBL14502222 0.78 NAAA (0.43) NAAALTA4HL3MBTL1ALDH1A1POLB
SCHEMBL20557014 0.77 TDP1 (0.51) LTA4HL3MBTL1ALDH1A1APPOPRM1
SCHEMBL16267407 0.77 CHRM5 (0.46) LTA4HL3MBTL1ALDH1A1POLBOPRM1
SCHEMBL27799490 0.77 TAAR1 (0.43) NAAAOPRM1OPRD1OPRK1TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5599966-A SUITABLE FOR TREATMENT OF DISEASES OF RESPIRATORY PASSAGES BYK NEDERLAND BV (NL) 1997-02-04 US disclosed
EP-0664788-A1 SUBSTITUTED ETHANOLAMINE ESTERS Byk Nederland BV (NL) 1995-08-02 EP disclosed
WO-1994008945-A1 SUBSTITUTED ETHANOLAMINE ESTERS BYK NEDERLAND BV (NL) 1994-04-28 WO disclosed